SCHEMBL6506347

SCHEMBL6506347

NC(=O)Nc1sc(NC(=O)c2ccc(-c3ccccc3)cc2)cc1C(N)=O

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 4/20 0.61
JAK2 O60674 2/20 0.61
JAK3 P52333 1/20 0.61
KDR P35968 1/20 0.56
PDCD1 Q15116 1/20 0.56
CD274 Q9NZQ7 1/20 0.56
MEN1 O00255 1/20 0.52
EIF2AK2 P19525 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
CHEK1 O14757 5/20 0.50
MAP4K4 O95819 1/20 0.50
NPC1 O15118 1/20 0.47
MAPT P10636 1/20 0.47
RAB9A P51151 1/20 0.47
PTPN5 P54829 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6530168 0.90 IKBKB (0.62) IKBKBJAK2JAK3KDRMEN1
SCHEMBL6509110 0.85 IKBKB (0.63) IKBKBJAK2JAK3KDRMEN1
SCHEMBL6530279 0.84 IKBKB (0.48) IKBKBJAK2JAK3KDRMEN1
SCHEMBL6507728 0.84 IKBKB (0.50) IKBKBJAK2JAK3KDRMEN1
SCHEMBL6508136 0.84 IKBKB (0.60) IKBKBJAK2JAK3MEN1EIF2AK2
SCHEMBL6512284 0.83 CHEK1 (0.47) IKBKBJAK2JAK3KDRMEN1
SCHEMBL6511724 0.82 MAPT (0.51) IKBKBJAK2JAK3KDRMEN1
SCHEMBL6514879 0.82 PARP10 (0.53) IKBKBKDRMEN1KMT2ACHEK1
SCHEMBL6505096 0.81 IKBKB (0.47) IKBKBJAK2JAK3MEN1EIF2AK2
SCHEMBL6509621 0.81 SMN1; SMN2 (0.65) IKBKBKDRMEN1KMT2ACHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005051381-A1 Substituted urea-octatydroindols as antagonists of melanin concentrating hormone receptor 1 (MCH1R) BIOVITRUM AB (SE) 2005-06-09 WO claimed
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed