SCHEMBL6528864

SCHEMBL6528864

COC(=O)c1c(CN2CCC(N3CCCCC3)CC2)c(-c2ccccc2)nc2ncc(Br)cc12

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 15/20 0.55
TACR3 P29371 6/20 0.55
TACR2 P21452 5/20 0.55
OPRM1 P35372 2/20 0.55
KCNH2 Q12809 2/20 0.51
OPRK1 P41145 1/20 0.49
CACNA1C Q13936 1/20 0.48
SCN5A Q14524 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6533888 0.91 TRPV4 (0.54) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL6506812 0.86 TRPV4 (0.58) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL5203642 0.85 TRPV4 (0.73) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL5202474 0.82 TACR3 (0.59) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL5945408 0.81 TRPV4 (0.55) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL6868096 0.79 TRPV4 (0.62) TRPV4TACR3TACR2KCNH2CACNA1C
SCHEMBL6853291 0.79 TRPV4 (0.55) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL2372637 0.79 TRPV4 (0.75) TRPV4TACR3TACR2KCNH2CACNA1C
SCHEMBL6506224 0.78 TACR3 (0.38) TACR3TACR2KCNH2OPRK1
SCHEMBL6393346 0.76 TRPV4 (0.58) TRPV4TACR3TACR2OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO disclosed