SCHEMBL6507356

SCHEMBL6507356

O=C(O)C1CCN(c2cccc(Cl)c2Cl)CC1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 10/20 0.83
DRD2 P14416 5/20 0.54
DRD3 P35462 4/20 0.54
ADRB1 P08588 1/20 0.54
RAB9A P51151 1/20 0.51
DRD4 P21917 1/20 0.51
GAA P10253 1/20 0.51
APAF1 O14727 1/20 0.50
NSD2 O96028 1/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
THRB P10828 1/20 0.50
CASP3 P42574 1/20 0.50
RECQL P46063 1/20 0.50
GALK1 P51570 1/20 0.50
KMT2A Q03164 1/20 0.50
HKDC1 Q2TB90 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31381185 1.00 NOTUM (0.83) NOTUMDRD2DRD3ADRB1RAB9A
SCHEMBL5800932 0.88 NOTUM (0.81) NOTUMADRB1RAB9AGAAAPAF1
SCHEMBL5800332 0.84 NOTUM (0.61) NOTUMRAB9AGAAAPAF1NSD2
SCHEMBL2555675 0.82 NOTUM (0.58) NOTUMRAB9AGAAAPAF1NSD2
SCHEMBL2558768 0.81 GAA (0.78) NOTUMRAB9AGAAAPAF1NSD2
SCHEMBL2939905 0.79 NOTUM (0.79) NOTUM
SCHEMBL27237946 0.79 DRD2 (0.60) NOTUMDRD2DRD3ADRB1DRD4
SCHEMBL31458523 0.79 TSHR (0.60) NOTUMGAAPOLBMAPTKMT2A
SCHEMBL2072056 0.77 NOTUM (0.83) NOTUMMAPTLMNAHTT
Maleic Acid SCHEMBL22720989 0.77 NOTUM (0.55) NOTUMDRD2DRD3ADRB1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250340557-A1 PYRIMIDINE DERIVATIVE ASKA PHARMACEUTICAL CO., LTD. (JP) 2025-11-06 US disclosed
EP-4570798-A1 AROMATIC HETEROCYCLIC CYCLOHEXYL AMINOALKYL PIPERIDINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF Jiangsu NHWA Pharmaceutical Co., Ltd (CN) 2025-06-18 EP disclosed
EP-4553068-A1 PYRIMIDINE DERIVATIVES ASKA Pharmaceutical Co., Ltd. (JP) 2025-05-14 EP disclosed
WO-2024032530-A1 AROMATIC HETEROCYCLIC CYCLOHEXYL AMINOALKYL PIPERIDINE DERIVATIVE, PREPARATION METHOD AND USE THEREOF 江苏恩华药业股份有限公司 2024-02-15 WO disclosed
WO-2024010015-A1 PYRIMIDINE DERIVATIVES あすか製薬株式会社 2024-01-11 WO disclosed
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250340557-A1 PYRIMIDINE DERIVATIVE PTGES, PTGS1, PTGIS NOTUM 2160/4885DRD2 2673/4885DRD3 3491/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.