SCHEMBL6508561

SCHEMBL6508561

CC(=O)N(c1ccc2ccc3cccc4ccc1c2c34)[C@@H](C)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
HPGD P15428 4/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 4/20 0.38
HSD17B10 Q99714 3/20 0.38
CYP1A2 P05177 3/20 0.38
MEN1 O00255 2/20 0.38
GLA P06280 1/20 0.38
POLB P06746 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP3A4 P08684 2/20 0.38
TSHR P16473 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
AKR1B1 P15121 2/20 0.36
SMPD2 O60906 1/20 0.36
GAA P10253 2/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6511954 0.82 ALDH1A1 (0.35) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL6511949 0.82 ALDH1A1 (0.35) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL6113112 0.81 SMPD2 (0.47) AKR1B1SMPD2GAA
SCHEMBL6119288 0.81 SMPD2 (0.47) AKR1B1SMPD2GAA
SCHEMBL6113113 0.81 SMPD2 (0.47) AKR1B1SMPD2GAA
SCHEMBL6517627 0.74 EPHX2 (0.38) KMT2A
N-Benzylmethylamine SCHEMBL9274090 0.70 L3MBTL1 (0.44) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL500318 0.69 ALDH1A1 (0.46) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL7776950 0.69 MEN1 (0.43) ALDH1A1KDM4EMAPTKMT2AMEN1
SCHEMBL16728481 0.69 MEN1 (0.43) ALDH1A1KDM4EMAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1585485-A2 COMPOSITIONS FOR THE REDUCTION OF HAIR GROWTH THE GILLETTE COMPANY (US) 2005-10-19 EP claimed
WO-2004064749-A2 COMPOSITIONS FOR THE REDUCTION OF HAIR GROWTH THE GILLETTE COMPANY (US) 2004-08-05 WO claimed
US-20040141935-A1 Reduction of hair growth GILLETTE COMPANY, THE 2004-07-22 US claimed
EP-4620463-A1 ACTIVE AGENT FOR USE IN HAIR GROWTH REGULATION CUTANEON - Skin & Hair Innovations GmbH (DE) 2025-09-24 EP disclosed
US-20230321122-A1 ACTIVE AGENT MODULATING THE ACTIVITY OF AN ION CHANNEL FOR USE IN HAIR GROWTH REGULATION CUTANEON SKIN & HAIR INNOVATIONS GMBH (DE) 2023-10-12 US disclosed
EP-3766545-B1 ACTIVE AGENT FOR USE IN HAIR GROWTH REGULATION CUTANEON SKIN & HAIR INNOVATIONS GMBH (DE) 2023-08-16 EP disclosed
WO-2022043171-A1 ACTIVE AGENT MODULATING THE ACTIVITY OF AN ION CHANNEL FOR USE IN HAIR GROWTH REGULATION MONASTERIUM LABORATORY SKIN & HAIR RESEARCH SOLUTIONS GMBH (DE) 2022-03-03 WO disclosed
EP-3960150-A1 ACTIVE AGENT MODULATING THE ACTIVITY OF AN ION CHANNEL FOR USE IN HAIR GROWTH REGULATION Monasterium Laboratory Skin & Hair Research Solutions GmbH (DE) 2022-03-02 EP disclosed
WO-2021009177-A1 ACTIVE AGENT FOR USE IN HAIR GROWTH REGULATION MONASTERIUM LABORATORY SKIN & HAIR RESEARCH SOLUTIONS GMBH (DE) 2021-01-21 WO disclosed
EP-3766545-A1 ACTIVE AGENT FOR USE IN HAIR GROWTH REGULATION Monasterium Laboratory Skin & Hair Research Solutions GmbH (DE) 2021-01-20 EP disclosed
US-20040141935-A1 Reduction of hair growth GILLETTE COMPANY, THE 2004-07-22 US disclosed