SCHEMBL6508770

SCHEMBL6508770

COC(=O)c1c(CBr)c(C#N)cc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.41
NCEH1 Q6PIU2 1/20 0.40
ALDH1A1 P00352 7/20 0.40
HPGD P15428 6/20 0.40
KDM4E B2RXH2 5/20 0.40
KDM5A P29375 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CRHBP P24387 2/20 0.40
CRHR2 Q13324 2/20 0.40
LMNA P02545 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AR P10275 1/20 0.37
PLA2G2A P14555 3/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 2/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603195 0.88 POLB (0.42) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL6608041 0.85 POLB (0.40) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL6604599 0.84 ALOX5 (0.42) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL4676934 0.81 MEN1 (0.45) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL6510652 0.81 NCEH1 (0.44) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL10699646 0.81 NCEH1 (0.44) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL6229441 0.80 ALDH1A1 (0.52) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL6603583 0.79 ALDH1A1 (0.42) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL6610048 0.78 NCEH1 (0.41) POLBNCEH1ALDH1A1HPGDKDM4E
SCHEMBL6603719 0.77 NCEH1 (0.40) POLBNCEH1ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO disclosed