SCHEMBL6509083

SCHEMBL6509083

C(=CN1CCOCC1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.54
ALDH1A1 P00352 9/20 0.48
ALOX15 P16050 1/20 0.48
TSHR P16473 1/20 0.48
MAOB P27338 1/20 0.47
LMNA P02545 1/20 0.47
HSP90AA1 P07900 2/20 0.46
MAPT P10636 5/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
NPC1 O15118 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
HPGD P15428 2/20 0.46
ALOX12 P18054 2/20 0.46
POLB P06746 2/20 0.46
USP2 O75604 1/20 0.46
MAPK1 P28482 1/20 0.46
PRKDC P78527 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6509077 1.00 RAB9A (0.54) RAB9AALDH1A1ALOX15TSHRMAOB
SCHEMBL28121251 0.88 RAB9A (0.47) RAB9AALDH1A1ALOX15TSHRMAOB
SCHEMBL5572239 0.84 MAOB (0.50) RAB9AALDH1A1MAOBLMNAMAPT
SCHEMBL28546334 0.84 MAOB (0.50) RAB9AALDH1A1MAOBLMNAMAPT
SCHEMBL11080877 0.82 RAB9A (0.55) RAB9AALDH1A1TSHRLMNAMAPT
SCHEMBL10410292 0.82 L3MBTL1 (0.55) RAB9AALDH1A1TSHRLMNAMAPT
SCHEMBL10410291 0.82 L3MBTL1 (0.55) RAB9AALDH1A1TSHRLMNAMAPT
SCHEMBL11080880 0.82 RAB9A (0.55) RAB9AALDH1A1TSHRLMNAMAPT
SCHEMBL6516804 0.80 KMT2A (0.48) RAB9AALDH1A1MAOBLMNAHSP90AA1
SCHEMBL6516806 0.80 KMT2A (0.48) RAB9AALDH1A1MAOBLMNAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005077885-A1 RUTHENIUM-CATALYZED HYDROAMINATION OF OLEFINS YALE UNIVERSITY (US) 2005-08-25 WO disclosed
EP-0558656-B1 NEW METHODS FOR THE CATALYTIC REDUCTION OF ORGANIC SUBSTRATES MASSACHUSETTS INST TECHNOLOGY (US) 1996-04-17 EP disclosed
EP-0558656-A1 NEW METHODS FOR THE CATALYTIC REDUCTION OF ORGANIC SUBSTRATES. MASSACHUSETTS INST TECHNOLOGY (US) 1993-09-08 EP disclosed
US-5220020-A Catalytic reduction of organic carbonyls using metal catalysts MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1993-06-15 US disclosed
WO-1992009545-A2 NEW METHODS FOR THE CATALYTIC REDUCTION OF ORGANIC SUBSTRATES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1992-06-11 WO disclosed
US-4486588-A Cyclohexadiene carboxylate insecticide intermediates FMC CORPORATION (US) 1984-12-04 US disclosed