SCHEMBL6509235

SCHEMBL6509235

NN(N)c1cccc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.52
ALDH1A1 P00352 3/20 0.48
TSHR P16473 2/20 0.48
HSD17B10 Q99714 2/20 0.48
CYP3A4 P08684 1/20 0.48
HPGD P15428 1/20 0.48
KEAP1 Q14145 1/20 0.48
CYP2A6 P11509 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
CYP1A2 P05177 2/20 0.42
HPRT1 P00492 2/20 0.42
HTR1B P28222 2/20 0.41
AOC3 Q16853 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4141823 0.85 SIGMAR1 (0.52) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL7067991 0.85 SIGMAR1 (0.52) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL29143191 0.81 SIGMAR1 (0.48) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL29495790 0.81 SIGMAR1 (0.59) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL3887404 0.81 SIGMAR1 (0.59) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL2575466 0.81 SIGMAR1 (0.53) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL6568773 0.79 SIGMAR1 (0.56) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL516020 0.79 SIGMAR1 (0.56) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL11672429 0.79 SIGMAR1 (0.56) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4
SCHEMBL29870751 0.79 SIGMAR1 (0.56) SIGMAR1ALDH1A1TSHRHSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013032284-A1 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUNDS AND ORGANIC ELECTROLUMINESCENT DEVICE USING THE SAME ROHM AND HAAS ELECTRONIC MATERIALS KOREA LTD. (KR) 2013-03-07 WO disclosed
EP-1499659-A1 NANOPARTICULATE ORGANIC UV ABSORBER BASF AKTIENGESELLSCHAFT (DE) 2005-01-26 EP disclosed
WO-2003085033-A1 NANOPARTICULATE ORGANIC UV ABSORBER BASF AKTIENGESELLSCHAFT (DE) 2003-10-16 WO disclosed
EP-0178960-B1 DIESEL FUEL COMPOSITIONS ETHYL PETROLEUM ADDITIVES, INC. (US) 1988-10-12 EP disclosed
US-4736015-A FROM DI-(ORTETRA) ESTER OF BENZHYDROL 3,3*,4,4*-TETRACARBOXYLIC ACID AND AROMATIC DIAMINE INSTITUT FRANCAIS DU PETROLE (FR) 1988-04-05 US disclosed
EP-0178960-A1 Diesel fuel compositions ETHYL PETROLEUM ADDITIVES, INC. (US) 1986-04-23 EP disclosed