SCHEMBL6510068

SCHEMBL6510068

CN(C(=O)O)C1CN(c2cc(-c3ccccc3)nc(N)n2)C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.55
HTR3A P46098 1/20 0.55
LMNA P02545 2/20 0.54
USP2 O75604 1/20 0.54
TSHR P16473 1/20 0.54
HTT P42858 1/20 0.54
HSD17B10 Q99714 1/20 0.54
SCN2A Q99250 1/20 0.47
HRH3 Q9Y5N1 3/20 0.46
AURKA O14965 1/20 0.45
PDPK1 O15530 1/20 0.45
AURKB Q96GD4 1/20 0.45
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPK10 P53779 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6023054 0.91 HTR3A (0.54) HRH4HTR3ALMNAUSP2TSHR
SCHEMBL605156 0.86 HRH3 (0.62) HRH4HTR3ALMNAUSP2TSHR
SCHEMBL23931281 0.82 PDPK1 (0.43) HRH4HTR3ALMNAUSP2TSHR
SCHEMBL1773838 0.80 LMNA (0.51) LMNAHTTHRH3AURKAPDPK1
SCHEMBL23931287 0.80 HRH3 (0.39) HRH4HTR3ALMNAUSP2TSHR
SCHEMBL6023493 0.79 JAK2 (0.45) HRH4HTR3ALMNAUSP2TSHR
Hydrochloric Acid SCHEMBL602600 0.79 HTR3A (0.58) HRH4HTR3ALMNAUSP2TSHR
SCHEMBL6512558 0.78 LMNA (0.56) HRH4HTR3ALMNAUSP2TSHR
SCHEMBL4420312 0.78 HRH3 (0.57) HRH4HRH3AURKAPDPK1AURKB
SCHEMBL1990283 0.78 HRH3 (0.48) HRH4LMNAHRH3AURKAPDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005054239-A1 2-AMINOPYRIMIDINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2005-06-16 WO disclosed