SCHEMBL6510104

SCHEMBL6510104

CC(=O)NCC(C)(C)C(=O)N1CCC(Oc2ncnc(Oc3ccc(S(C)(=O)=O)cc3F)c2C)CC1

nearest known ligand 0.68

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 20/20 0.68
CYP2C9 P11712 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2401945 0.85 GPR119 (0.70) GPR119CYP2C9
SCHEMBL2786447 0.85 GPR119 (0.79) GPR119CYP2C9
SCHEMBL2401493 0.85 GPR119 (0.66) GPR119CYP2C9
SCHEMBL5070635 0.84 GPR119 (0.64) GPR119CYP2C9
SCHEMBL386489 0.83 GPR119 (0.74) GPR119CYP2C9
SCHEMBL390259 0.83 GPR119 (0.74) GPR119CYP2C9
SCHEMBL390528 0.83 GPR119 (0.69) GPR119CYP2C9
SCHEMBL389216 0.83 GPR119 (0.74) GPR119CYP2C9
SCHEMBL388993 0.83 GPR119 (0.74) GPR119CYP2C9
SCHEMBL388992 0.83 GPR119 (0.74) GPR119CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050070562-A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto ARENA PHARMACEUTICALS, INC. 2005-03-31 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050070562-A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto CYP7A1, CYP27A1, SULT2A1 GPR119 13/4885CYP2C9 56/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.