SCHEMBL6510295

SCHEMBL6510295

COc1ccc(OC)c(Sc2ncccc2C(=O)NC(CC(=O)O)c2ccc(NC(=O)c3c(Cl)cncc3Cl)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.43
ITGB1 P05556 4/20 0.42
ITGA4 P13612 4/20 0.42
CTSA P10619 9/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HPGD P15428 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ATP4A P20648 1/20 0.39
ATP4B P51164 1/20 0.39
THRB P10828 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6510654 0.94 ITGB1 (0.48) LMNAITGB1ITGA4CTSAALDH1A1
SCHEMBL6514009 0.79 ITGB1 (0.58) ITGB1ITGA4ALDH1A1SMN1; SMN2MEN1
SCHEMBL6518236 0.77 ITGB1 (0.52) LMNAITGB1ITGA4CTSASMN1; SMN2
SCHEMBL6512426 0.76 ITGB1 (0.53) ITGB1ITGA4ALDH1A1SMN1; SMN2MEN1
SCHEMBL6509549 0.74 ITGB1 (0.63) ITGB1ITGA4CTSA
SCHEMBL6514203 0.72 ITGB1 (0.49) LMNAITGB1ITGA4ALDH1A1SMN1; SMN2
SCHEMBL6518082 0.71 ITGB1 (0.57) ITGB1ITGA4
SCHEMBL6513196 0.70 ITGB1 (0.53) ITGB1ITGA4KMT2A
SCHEMBL6512467 0.70 ALDH1A1 (0.60) LMNAALDH1A1KDM4ESMN1; SMN2HPGD
SCHEMBL6513291 0.70 ITGB1 (0.48) ITGB1ITGA4SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953798-B1 β-alanine derivates CELLTECH R&D LIMITED (GB) 2005-10-11 US claimed
EP-1135371-A1 BETA-ALANINE DERIVATIVES AS ALPHA 4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2001-09-26 EP claimed
WO-2000032575-A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2000-06-08 WO claimed
US-6953798-B1 β-alanine derivates CELLTECH R&D LIMITED (GB) 2005-10-11 US disclosed