SCHEMBL6513439

SCHEMBL6513439

COc1nc(NCCO)nc(NC(CC(=O)O)c2ccc(NC(=O)c3c(Cl)cncc3Cl)cc2)n1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.72
ITGA4 P13612 18/20 0.72
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6517093 0.93 ITGB1 (0.70) ITGB1ITGA4ALDH1A1HPGDSMN1; SMN2
SCHEMBL5364460 0.84 ITGB1 (1.00) ITGB1ITGA4
SCHEMBL7449206 0.79 ITGB1 (0.91) ITGB1ITGA4
SCHEMBL7104241 0.78 ITGB1 (0.51) ITGB1ITGA4
SCHEMBL7104244 0.78 ITGB1 (0.51) ITGB1ITGA4
SCHEMBL5368089 0.77 ITGB1 (1.00) ITGB1ITGA4
SCHEMBL7263470 0.76 ITGB1 (0.69) ITGB1ITGA4
SCHEMBL7263468 0.76 ITGB1 (0.69) ITGB1ITGA4
SCHEMBL6518236 0.75 ITGB1 (0.52) ITGB1ITGA4SMN1; SMN2
SCHEMBL6509549 0.75 ITGB1 (0.63) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953798-B1 β-alanine derivates CELLTECH R&D LIMITED (GB) 2005-10-11 US claimed
EP-1135371-A1 BETA-ALANINE DERIVATIVES AS ALPHA 4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2001-09-26 EP claimed
WO-2000032575-A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2000-06-08 WO claimed
US-6953798-B1 β-alanine derivates CELLTECH R&D LIMITED (GB) 2005-10-11 US disclosed
EP-1135371-A1 BETA-ALANINE DERIVATIVES AS ALPHA 4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2001-09-26 EP disclosed
WO-2000032575-A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS CELLTECH THERAPEUTICS LIMITED (GB) 2000-06-08 WO disclosed