SCHEMBL6513644

SCHEMBL6513644

CCCCCOc1cccc(N=C(N)Nc2cccc(C)c2)c1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.64
GRIN2D O15399 5/20 0.64
GRIN3B O60391 5/20 0.64
GRIN1 Q05586 5/20 0.64
GRIN2A Q12879 5/20 0.64
GRIN2B Q13224 5/20 0.64
GRIN2C Q14957 5/20 0.64
GRIN3A Q8TCU5 5/20 0.64
FAAH O00519 1/20 0.50
THRB P10828 1/20 0.48
NR1H4 Q96RI1 2/20 0.47
CYP1A2 P05177 1/20 0.47
POLB P06746 1/20 0.47
CYP2D6 P10635 1/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
MAPK1 P28482 1/20 0.46
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4985390 0.93 SIGMAR1 (0.64) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6720704 0.82 SIGMAR1 (0.86) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL5923034 0.81 THRB (0.54) FAAHTHRBNR1H4MAPK1TSHR
SCHEMBL6422901 0.80 SIGMAR1 (1.00) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6512853 0.80 SIGMAR1 (0.72) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6717633 0.79 SIGMAR1 (0.86) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL27003088 0.76 SIGMAR1 (0.85) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9858310 0.75 NR1H4 (0.68) FAAHTHRBNR1H4
SCHEMBL6720947 0.75 SIGMAR1 (0.85) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6720803 0.75 SIGMAR1 (1.00) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005095345-A2 HETEROARYL GUANIDINES AS INHIBITORS OF VIRAL REPLICATION ACHILLION PHARMACEUTICALS, INC. (US) 2005-10-13 WO claimed