SCHEMBL6524693

SCHEMBL6524693

N[C@@H]1CCN(C(=O)OCc2ccccc2)C1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.67
CYP2C19 P33261 1/20 0.67
NPC1 O15118 2/20 0.66
RAB9A P51151 2/20 0.66
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
GRIN2B Q13224 9/20 0.53
HTT P42858 1/20 0.53
CYP2D6 P10635 4/20 0.52
CYP2C9 P11712 4/20 0.52
PDE4B Q07343 1/20 0.50
USP30 Q70CQ3 1/20 0.49
CYP3A4 P08684 3/20 0.49
ENPP2 Q13822 1/20 0.48
F13A1 P00488 1/20 0.47
TGM2 P21980 1/20 0.47
TGM1 P22735 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1189968 1.00 SMN1; SMN2 (0.67) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
SCHEMBL266047 1.00 SMN1; SMN2 (0.67) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL716733 0.99 SMN1; SMN2 (0.65) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL2514584 0.99 SMN1; SMN2 (0.65) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL6175666 0.99 SMN1; SMN2 (0.65) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
Acetic Acid SCHEMBL2495069 0.96 SMN1; SMN2 (0.62) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
Trifluoroacetic Acid SCHEMBL952417 0.92 SMN1; SMN2 (0.58) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
SCHEMBL764193 0.92 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
SCHEMBL654999 0.92 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19NPC1RAB9AMEN1
SCHEMBL12791106 0.92 SMN1; SMN2 (0.60) SMN1; SMN2CYP2C19NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802500-B1 MELANOCORTIN SUBTYPE-2 RECEPTOR (MC2R) ANTAGONISTS AND USES THEREOF CRINETICS PHARMACEUTICALS INC (US) 2026-05-27 EP disclosed
US-20260132140-A1 IMIDAZOLYL-AMINO-PYRAZINE-CARBONITRILS AS CHK-1 INHIBITORS BENEVOLENTAI BIO LTD (GB) 2026-05-14 US disclosed
EP-4720058-A2 BIFUNCTIONAL DEGRADERS AND USES THEREOF Casma Therapeutics, Inc. (US) 2026-04-08 EP disclosed
US-12479825-B2 Melanocortin subtype-2 receptor (MC2R) antagonists and uses thereof Crinetics Pharmaceuticals, Inc. (US) 2025-11-25 US disclosed
US-12479828-B2 Melanocortin subtype-2 receptor (MC2R) antagonists and uses thereof Crinetics Pharmaceuticals, Inc. (US) 2025-11-25 US disclosed
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2025-08-05 US disclosed
EP-4590671-A1 IMIDAZOLYL-AMINO-PYRAZINE-CARBONITRILS AS CHK-1 INHIBITORS BenevolentAI Bio Limited (GB) 2025-07-30 EP disclosed
WO-2024249291-A2 BIFUNCTIONAL DEGRADERS AND USES THEREOF CASMA THERAPEUTICS, INC. (US) 2024-12-05 WO disclosed
CN-112533904-B Melanocortin subtype-2 receptor (MC 2R) antagonists and uses thereof 克林提克斯医药股份有限公司 2024-10-29 CN disclosed
US-20240300920-A1 MELANOCORTIN SUBTYPE-2 RECEPTOR (MC2R) ANTAGONISTS AND USES THEREOF Crinetics Pharmaceuticals, Inc. 2024-09-12 US disclosed
US-7786312-B2 Methods of preparing heterocyclic boronic acids and derivatives thereof PHENOMIX CORPORATION (US) 2010-08-31 US disclosed
CN-101239937-B Method for preparing optical activity R-(-)-1-benzylcarbonyl-3-aminopyrrolidine and hydrochloride thereof SHANGHAI ABA CHEMICALS CO LTD 2010-05-19 CN disclosed
US-20100087658-A1 METHODS AND INTERMEDIATES FOR SYNTHESIS OF SELECTIVE DPP-IV INHIBITORS PHENOMIX CORPORATION (US) 2010-04-08 US disclosed
CN-101679238-A methods and intermediates for synthesis of selective dpp-iv inhibitors PHENOMIX CORP 2010-03-24 CN disclosed
US-20080300413-A1 Methods of Preparing Hetercyclic Boronic Acids and Derivatives Thereof SINO-MED INTERNATIONAL ALLIANCE, INC. 2008-12-04 US disclosed
US-20080300413-A1 Methods of Preparing Hetercyclic Boronic Acids and Derivatives Thereof SINO-MED INTERNATIONAL ALLIANCE, INC. 2008-12-04 US disclosed
WO-2008109681-A2 METHODS AND INTERMEDIATES FOR SYNTHESIS OF SELECTIVE DPP-IV INHIBITORS PHENOMIX CORPORATION (US) 2008-09-12 WO disclosed
CN-101239937-A Method for preparing optical activity R-(-)-1-benzylcarbonyl-3-aminopyrrolidine and hydrochloride thereof SHANGHAI ABA CHEMICALS CO LTD (CN) 2008-08-13 CN disclosed
US-6331548-B1 PREVENTION OR TREATMENT OF CYTOKINE RELATED DISEASES SUNTORY LIMITED (JP) 2001-12-18 US disclosed
EP-0978516-A1 1-CYCLOALKYL-1,8-NAPHTHYRIDIN-4-ONE DERIVATIVES WITH PHOSPHODIESTERASE IV INHIBITORY ACTIVITY SUNTORY LIMITED (JP) 2000-02-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080300413-A1 Methods of Preparing Hetercyclic Boronic Acids and Derivatives Thereof HLCS, NISCH, BTD SMN1; SMN2 2610/4885CYP2C19 389/4885NPC1 1901/4885
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors MERTK, RET, ERBB2 SMN1; SMN2 2563/4885CYP2C19 637/4885NPC1 649/4885
US-20100087658-A1 METHODS AND INTERMEDIATES FOR SYNTHESIS OF SELECTIVE DPP-IV INHIBITORS DPP4, DPP3, DPP7 SMN1; SMN2 3932/4885CYP2C19 2245/4885NPC1 2124/4885
US-20260132140-A1 IMIDAZOLYL-AMINO-PYRAZINE-CARBONITRILS AS CHK-1 INHIBITORS CHEK1, CHEK2, BUB1 SMN1; SMN2 2599/4885CYP2C19 3969/4885NPC1 1573/4885
US-12479825-B2 Melanocortin subtype-2 receptor (MC2R) antagonists and uses thereof MC3R, MC1R, MC2R SMN1; SMN2 2938/4885CYP2C19 1504/4885NPC1 1729/4885
US-20240300920-A1 MELANOCORTIN SUBTYPE-2 RECEPTOR (MC2R) ANTAGONISTS AND USES THEREOF MC3R, MC1R, MC2R SMN1; SMN2 2938/4885CYP2C19 1504/4885NPC1 1729/4885
US-12479828-B2 Melanocortin subtype-2 receptor (MC2R) antagonists and uses thereof MC3R, MC1R, MC2R SMN1; SMN2 2938/4885CYP2C19 1504/4885NPC1 1729/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.