SCHEMBL6526696

SCHEMBL6526696

COC(=O)CC(=O)C=Cc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 1/20 0.66
MAPT P10636 4/20 0.60
APP P05067 1/20 0.60
GSK3B P49841 2/20 0.59
ALDH1A1 P00352 4/20 0.56
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
KDM4E B2RXH2 1/20 0.55
RAB9A P51151 1/20 0.55
KCNH2 Q12809 1/20 0.55
BACE1 P56817 2/20 0.54
GLA P06280 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
HDAC3 O15379 2/20 0.52
HDAC4 P56524 2/20 0.52
HDAC1 Q13547 2/20 0.52
HDAC2 Q92769 2/20 0.52
HDAC8 Q9BY41 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
TNKS O95271 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10348533 1.00 HAO1 (0.66) HAO1MAPTAPPGSK3BALDH1A1
SCHEMBL27435225 0.92 HAO1 (0.60) HAO1MAPTAPPGSK3BALDH1A1
SCHEMBL316674 0.87 HAO1 (0.84) HAO1MAPTAPPGSK3BALDH1A1
SCHEMBL3439644 0.87 HAO1 (0.84) HAO1MAPTAPPGSK3BALDH1A1
SCHEMBL3105207 0.86 HAO1 (0.62) HAO1MAPTAPPGSK3BALDH1A1
SCHEMBL3105202 0.86 HAO1 (0.62) HAO1MAPTAPPGSK3BALDH1A1
Dimethylamine SCHEMBL14875132 0.85 HAO1 (0.75) HAO1MAPTAPPGSK3BALDH1A1
SCHEMBL8467852 0.84 AKR1B1 (0.76) GSK3BBACE1MAOBAKR1B10AKR1B1
SCHEMBL6954034 0.83 BACE1 (0.55) MAPTAPPGSK3BALDH1A1MEN1
SCHEMBL10759485 0.83 GSK3B (0.60) MAPTGSK3BALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0239105-B1 PHARMACEUTICAL COMPOSITIONS CONTAINING 5-PHENYL-1,3-DIOXOALKENYL COMPOUNDS G.D. Searle & Co. (US) 1990-05-23 EP claimed
EP-0239105-A2 Pharmaceutical compositions containing 5-phenyl-1,3-dioxoalkenyl compounds G.D. Searle & Co. (US) 1987-09-30 EP claimed
US-20050209117-A1 Complexing agent for treating metallic and plastic surfaces BASF AKTIENGESELLSCHAFT (DE) 2005-09-22 US disclosed
EP-1023267-B1 PYRIDYL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CERMOL SA (CH) 2003-09-17 EP disclosed
US-6482841-B1 Pyridyl compounds and pharmaceutical compositions containing them CERMOL S.A. (CH) 2002-11-19 US disclosed
EP-1023267-A1 PYRIDYL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 2000-08-02 EP disclosed
US-5951841-A ACIDIC ELECTROPLATING BATHS COMPRISING BRIGHTENERS FOR THE ELECTROLYTIC DEPOSITION OF METALLIC INORGANIC LAYERS ONTO SHAPED ARTICLES BASF AKTIENGESELLSCHAFT (DE) 1999-09-14 US disclosed
WO-1999019302-A1 PYRIDYL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CERMOL S.A. (CH) 1999-04-22 WO disclosed
US-5421990-A An acidic aqueous electrodeposition bath having a nontoxic, nonirritating brightener comprising a benzylidine malonic ester or acetylacetonate BASF AKTIENGESELLSCHAFT (DE) 1995-06-06 US disclosed
EP-0239105-B1 PHARMACEUTICAL COMPOSITIONS CONTAINING 5-PHENYL-1,3-DIOXOALKENYL COMPOUNDS G.D. Searle & Co. (US) 1990-05-23 EP disclosed
US-4898877-A ANTIARRHYTHMIA AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1990-02-06 US disclosed
US-3951994-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-20 US disclosed
US-3948923-A HYPOTENSIVE, VASODILATION BAYER AKTIENGESELLSCHAFT (DT) 1976-04-06 US disclosed
US-3946026-A HYPOTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-03-23 US disclosed
US-3946028-A HYPOTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-03-23 US disclosed
US-3946027-A HYPOTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-03-23 US disclosed
US-3943140-A HYPOTENSIVE, VASODILATION BAYER AKTIENGESELLSCHAFT (DT) 1976-03-09 US disclosed
US-3939171-A HYPOTENSIVE, VASODILATION BAYER AKTIENGESELLSCHAFT (DT) 1976-02-17 US disclosed
US-3935220-A VASODILATION, HYPOTENSIVE BAYER AKTIENGESELLSCHAFT (DT) 1976-01-27 US disclosed
US-3935223-A 2-Amino-1,4-dihydropyridine derivatives BAYER AKTIENGESELLSCHAFT (DT) 1976-01-27 US disclosed