SCHEMBL6527189

SCHEMBL6527189

COc1c(N2CCC(C(O)C(F)(F)CO)C2)ccc2c(=O)c(C(=O)O)c(F)n(C3CC3)c12

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.50
CYP3A4 P08684 1/20 0.38
POLB P06746 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PRKD3 O94806 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
OPRM1 P35372 1/20 0.32
CLK2 P49760 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
LIPG Q9Y5X9 4/20 0.32
LIPC P11150 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320087 0.80 KCNH2 (0.50) KCNH2CYP3A4POLBKDM4EPRKD3
SCHEMBL5725020 0.75 KCNH2 (0.44) KCNH2CYP3A4POLBKDM4EPRKD3
SCHEMBL4370115 0.74 KCNH2 (0.41) KCNH2CYP3A4POLBKDM4EPRKD3
SCHEMBL4371545 0.71 KCNH2 (0.43) KCNH2CYP3A4KDM4E
SCHEMBL6489214 0.71 KCNH2 (0.74) KCNH2POLBKDM4EPRKD3ALDH1A1
SCHEMBL6377878 0.69 KCNH2 (0.75) KCNH2CYP3A4POLBKDM4EPRKD3
SCHEMBL9867308 0.68 PIM1 (0.45) KCNH2CYP3A4POLBPRKD3ALDH1A1
SCHEMBL8540093 0.67 KCNH2 (0.41) KCNH2POLBKDM4EPRKD3ALDH1A1
SCHEMBL140764 0.67 KCNH2 (0.37) KCNH2POLBKDM4EPRKD3ALDH1A1
SCHEMBL6378744 0.67 KCNH2 (0.44) KCNH2CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005026165-A1 QUINOLONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2005-03-24 WO claimed