SCHEMBL6527780

SCHEMBL6527780

CN1CCN(C2CCCc3ccc(O)cc32)CC1.CN1CCN(C2CCCc3ccc(OC(=O)c4ccc(N5CCOCC5)nc4)cc32)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 8/20 0.44
ADRA1A P35348 3/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MTNR1A P48039 4/20 0.38
FKBP1A P62942 1/20 0.38
HRH3 Q9Y5N1 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6406680 0.96 MTNR1B (0.47) MTNR1BADRA1ACNR1CNR2ALDH1A1
SCHEMBL6409730 0.80 CNR1 (0.54) CNR1CNR2
SCHEMBL6406808 0.77 CNR2 (0.51) CNR1CNR2
SCHEMBL6405341 0.73 MTNR1B (0.50) MTNR1B
SCHEMBL6403876 0.72 ADRA1D (0.46) MTNR1BADRA1ACNR1CNR2HRH3
SCHEMBL6405239 0.68 MTNR1B (0.55) MTNR1BCNR1CNR2ALOX15HSD17B10
SCHEMBL6404873 0.67 MTNR1B (0.52) MTNR1BCNR1CNR2ALDH1A1MTNR1A
SCHEMBL6001623 0.67 MTNR1B (0.70) MTNR1BMTNR1A
SCHEMBL22411069 0.66 MTNR1B (0.51) MTNR1BCNR1CNR2ALDH1A1KDM4E
SCHEMBL6403250 0.66 MTNR1B (0.48) MTNR1BCNR1CNR2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005113527-A1 TETRAHYDRONAPHTHYL- PIPERAZINES AS 5-HT1B ANTAGONISTS, INVERSE AGONISTS AND PARTIAL AGONISTS PFIZER PRODUCTS INC. (US) 2005-12-01 WO disclosed