SCHEMBL6506224

SCHEMBL6506224

COC(=O)c1c(C[N+]2(N3CCCCC3)CCCCC2)c(-c2ccccc2)nc2ncc(Br)cc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 6/20 0.38
KCNH2 Q12809 5/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
GABRA5 P31644 2/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA3 P34903 1/20 0.36
DHODH Q02127 1/20 0.35
PTGFR P43088 3/20 0.35
OPRK1 P41145 1/20 0.34
TACR2 P21452 2/20 0.34
MAPK8 P45983 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CNR1 P21554 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528864 0.78 TRPV4 (0.55) TACR3KCNH2OPRK1TACR2
SCHEMBL6533888 0.68 TRPV4 (0.54) TACR3KCNH2TACR2
SCHEMBL6506852 0.65 DHODH (0.56) TACR3GABRA5GABRA1GABRG2GABRB3
SCHEMBL2372430 0.64 TACR3 (0.50) TACR3KCNH2MAPTTACR2SMN1; SMN2
SCHEMBL6506812 0.63 TRPV4 (0.58) TACR3KCNH2TACR2
SCHEMBL28398501 0.63 AXL (0.48) GAAMAPTGABRA5GABRA1GABRG2
SCHEMBL2372595 0.63 SMN1; SMN2 (0.54) TACR3MAPTDHODHTACR2SMN1; SMN2
SCHEMBL5202872 0.61 HPGD (0.52) GAAMAPTDHODHPTGFRSMN1; SMN2
SCHEMBL5908880 0.61 KDM4E (0.48) GAAMAPTDHODHPTGFRSMN1; SMN2
SCHEMBL27729454 0.61 LMNA (0.53) TACR3MAPTDHODHTACR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO disclosed