SCHEMBL6528896

SCHEMBL6528896

C=CCN(CC=C)S(=O)(=O)CC=C

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16701357 0.91 KDM4E (0.33) KDM4EPOLBTDP1
SCHEMBL11873651 0.83 KDM4E (0.31) KDM4EPOLBTDP1
SCHEMBL27783120 0.81 RAB9A (0.44) KDM4EPOLBTDP1MEN1KMT2A
SCHEMBL11833468 0.77 KDM4E (0.35) KDM4EPOLBTDP1MEN1KMT2A
SCHEMBL2489037 0.75 ALDH1A1 (0.32) MEN1KMT2AALDH1A1
SCHEMBL11031928 0.75 KDM4E (0.39) KDM4EPOLBTDP1MEN1KMT2A
SCHEMBL973944 0.75 KDM4E (0.39) KDM4EPOLBTDP1MEN1KMT2A
SCHEMBL8652753 0.75 KDM4E (0.39) KDM4EPOLBTDP1MEN1KMT2A
SCHEMBL7239582 0.73
SCHEMBL6431047 0.72 KDM4E (0.38) KDM4EPOLBTDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104987330-A HETEROARYL PIPERIDINE AND HETEROARYL PIPERAZINE DERIVATIVES AS FUNGICIDES BAYER IP GMBH 2015-10-21 CN claimed
CN-103492380-A Heteroarylpiperidine and piperazine derivatives as fungicides BAYER IP GMBH 2014-01-01 CN claimed
CN-102414175-A Insecticidal arylpyrrolidines BAYER CROPSCIENCE AG 2012-04-11 CN claimed
CN-101663289-A Piperazinyl-propyl-pyrazole derivatives and the pharmaceutical composition that comprises them as dopamine d 4 receptor antagonists KOREA RES INST CHEM TECH 2010-03-03 CN claimed
CN-100400519-C N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines FMC CORP (DE) 2008-07-09 CN claimed
CN-101139340-A N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines BAYER CROPSCIENCE AG (US) 2008-03-12 CN claimed
CN-1729178-A N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines FMC CORP (US) 2006-02-01 CN claimed
CN-1196692-C Substituted benzopyran derivatives for the treatment of inflammation SEARLE & CO (US) 2005-04-13 CN claimed
CN-1105106-C Naphthol derivatives and process for preparation thereof UENO SEIYAKU OYO KENKYUJO KK (JP) 2003-04-09 CN claimed
CN-1317004-A Benzoyl derivatives, process for their preparation and their use as herbicides and plant growth regulators HOECHST SCHERING AGREVO GMBH (DE) 2001-10-10 CN claimed
CN-1208439-A Process for the preparation of substituted aryl lactic acid containing cyclodepsipeptides with 24 ring atoms BAYER AG (DE) 1999-02-17 CN claimed
CN-1157619-A Pyrimido [5-4-d] pyrimidines, drugs containing these compounds, their use and process for preparing them THOMAE GMBH DR K (DE) 1997-08-20 CN claimed
CN-1046898-A 1-Aryimidazole insecticides RHONE POULENC AGROCHIMIE (FR) 1990-11-14 CN claimed
CN-87103552-A Adopt malonate derivative to improve crop yield 1988-07-06 CN claimed
CN-104987330-A HETEROARYL PIPERIDINE AND HETEROARYL PIPERAZINE DERIVATIVES AS FUNGICIDES BAYER IP GMBH 2015-10-21 CN disclosed
CN-102596933-B Herbicidal pyrimidone derivatives DU PONT 2014-09-17 CN disclosed
CN-101663289-B Piperazinyl-propyl-pyrazole derivatives as dopamine d4 receptor antagonists, and pharmaceutical compositions containing the same KOREA RES INST CHEM TECH 2014-07-23 CN disclosed
EP-0286346-A2 Insecticidal substituted indazoles E.I. DU PONT DE NEMOURS AND COMPANY (US) 1988-10-12 EP disclosed
CN-87103552-A Adopt malonate derivative to improve crop yield 1988-07-06 CN disclosed
CN-85105723-A Herbicidal compositions containing 1-aryl-4-substituted-1, 4-dihydro-5H-tetrazol-5-ones and their sulfur analogs 1986-05-10 CN disclosed