SCHEMBL6530160

SCHEMBL6530160

CN(C)Cc1ccc(-c2cc(Nc3ccc4c(cnn4C)c3)ncn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.47
CYP1A2 P05177 4/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
MAPK1 P28482 2/20 0.43
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
GLA P06280 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ADORA2A P29274 1/20 0.43
TRPM5 Q9NZQ8 1/20 0.40
LMNA P02545 1/20 0.40
BACE1 P56817 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6531053 0.78 ROCK2 (0.46) CDC7CYP1A2CYP2D6CYP2C9CLK4
SCHEMBL6529438 0.71 CLK4 (0.43) CDC7CYP1A2CYP2D6CYP2C9CLK4
SCHEMBL22595054 0.71 CCNT1 (0.48) ABL1BCRSLC2A1
SCHEMBL26028314 0.68 EGFR (0.47) JAK1JAK3JAK2
SCHEMBL6531231 0.68 ROCK2 (0.47) ADORA2AJAK3IRAK4
SCHEMBL30728059 0.67 CDC7 (0.64) CDC7CYP1A2MAPK1ALDH1A1TRPM5
SCHEMBL15344154 0.66 TRPA1 (0.46) CDC7TRPM5
SCHEMBL4114729 0.66 USP2 (0.62) CYP1A2CYP2D6CLK4USP2ALDH1A1
SCHEMBL15189081 0.66 CDC7 (0.56) CDC7CYP1A2ALDH1A1ALOX15HSD17B10
SCHEMBL4103830 0.65 CCNT1 (0.55) CYP1A2CYP2D6CYP2C9CLK4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005103036-A1 PYRIMIDIN-4-YL-1H-INDAZOL-5YL-AMINES AS CHK1 KINASES INHIBITORS BIOFOCUS DISCOVERY LTD (GB) 2005-11-03 WO claimed