SCHEMBL6530243

SCHEMBL6530243

Nc1cccnc1NCCN1CCOCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
CYP1A2 P05177 6/20 0.50
CYP3A4 P08684 6/20 0.50
CYP2D6 P10635 6/20 0.50
LMNA P02545 5/20 0.50
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
HIF1A Q16665 3/20 0.50
ELANE P08246 1/20 0.50
CLK4 Q9HAZ1 1/20 0.49
TOP2A P11388 1/20 0.49
HSD17B10 Q99714 3/20 0.48
TDP1 Q9NUW8 3/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20966396 0.92 TSHR (0.53) KDM4ENPC1RAB9ACYP3A4CYP2D6
SCHEMBL6528467 0.83 L3MBTL1 (0.53) KDM4EL3MBTL1NPC1RAB9ACYP1A2
SCHEMBL28282944 0.81 KDM4E (0.59) KDM4EL3MBTL1NPC1RAB9AELANE
SCHEMBL6527214 0.78 MAPT (0.58) KDM4EL3MBTL1NPC1RAB9ACYP1A2
SCHEMBL20689339 0.77 ELANE (0.48) KDM4EL3MBTL1NPC1RAB9ACYP1A2
SCHEMBL11710830 0.77 FGFR1 (0.46)
SCHEMBL6528435 0.77 KMT2A (0.51) KDM4EL3MBTL1LMNAMEN1KMT2A
SCHEMBL29504400 0.77 KMT2A (0.51) KDM4EL3MBTL1LMNAMEN1KMT2A
SCHEMBL11263883 0.77 ALDH1A1 (0.45) KDM4ENPC1RAB9AHSD17B10ALDH1A1
SCHEMBL11235791 0.76 CYP3A4 (0.48) L3MBTL1NPC1RAB9ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107750251-A Isoxazolyl-substituted imidazopyridines 塞尔森瑞科有限责任公司 2018-03-02 CN disclosed
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed