SCHEMBL28282944

SCHEMBL28282944

NC(=O)c1cccnc1NCCN1CCOCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.59
ALDH1A1 P00352 3/20 0.59
HPGD P15428 1/20 0.59
HSD17B10 Q99714 1/20 0.59
L3MBTL1 Q9Y468 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
ELANE P08246 1/20 0.48
APAF1 O14727 1/20 0.48
MITF O75030 1/20 0.48
CASP7 P55210 1/20 0.48
CASP9 P55211 1/20 0.48
CASP6 P55212 1/20 0.48
CASP8 Q14790 1/20 0.48
MAPT P10636 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
HPGDS O60760 1/20 0.47
AURKA O14965 1/20 0.47
RPS6KB1 P23443 1/20 0.47
PARP1 P09874 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13701710 0.85 ADRA1D (0.58) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL13702259 0.84 CHIA (0.51) ALDH1A1ELANEMAPTSMN1; SMN2HPGDS
SCHEMBL13702335 0.82 ADRA1D (0.49) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL6402609 0.82 DRD2 (0.52) SMN1; SMN2
SCHEMBL6530243 0.81 KDM4E (0.52) KDM4EALDH1A1HPGDHSD17B10L3MBTL1
SCHEMBL11465420 0.80 ALDH1A1 (0.66) KDM4EALDH1A1HPGDPARP1PARP2
SCHEMBL11158275 0.79 MMP12 (0.50) ALDH1A1HSD17B10L3MBTL1NPC1RAB9A
SCHEMBL5947803 0.79 SMN1; SMN2 (0.51) ALDH1A1HPGDMAPTSMN1; SMN2HPGDS
SCHEMBL28870897 0.79 ALDH1A1 (0.53) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL4708251 0.78 GAA (0.50) KDM4EALDH1A1AURKARPS6KB1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061967-B The nicotinamide compounds replaced through heteroaryl 百时美施贵宝公司 2019-04-19 CN claimed