SCHEMBL6530478

SCHEMBL6530478

COc1ccc(Sc2nc(Nc3cccc(F)c3)nc(N[C@@H](CC(C)C)C(=O)NCCC3CCCN3C)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.43
CHRM3 P20309 8/20 0.39
CTSS P25774 5/20 0.39
CTSL P07711 4/20 0.39
ACKR3 P25106 2/20 0.36
ACP1 P24666 1/20 0.35
KCNH3 Q9ULD8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528788 0.89 CTSK (0.43) CTSKCTSSCTSLKCNH3
SCHEMBL6531499 0.85 PDPK1 (0.45) CTSK
SCHEMBL6530210 0.84 NPC1 (0.45) CTSK
SCHEMBL6530634 0.83 CTSK (0.45) CTSKCTSSCTSLKCNH3
SCHEMBL6528746 0.82 CTSK (0.44) CTSKCTSSCTSLKCNH3
SCHEMBL6531457 0.82 ATM (0.45) CTSKCTSSCTSLKCNH3
SCHEMBL6532662 0.81 CTSK (0.42) CTSKCTSSCTSLKCNH3
SCHEMBL6508189 0.81 KCNH3 (0.41) CTSKKCNH3
SCHEMBL6528931 0.81 KCNH3 (0.41) CTSKKCNH3
SCHEMBL6508192 0.81 KCNH3 (0.41) CTSKKCNH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO claimed
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed