SCHEMBL6531499

SCHEMBL6531499

COc1ccc(Sc2nc(Nc3cccc(F)c3)nc(N[C@@H](CC(C)C)C(=O)NCCN3CCOCC3)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.45
CTSK P43235 2/20 0.42
TSHR P16473 1/20 0.41
RECQL P46063 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
RAF1 P04049 1/20 0.40
BRAF P15056 1/20 0.40
POLB P06746 3/20 0.39
TACR2 P21452 3/20 0.39
GSK3A P49840 2/20 0.39
GSK3B P49841 1/20 0.39
RAB9A P51151 1/20 0.39
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528788 0.94 CTSK (0.43) PDPK1CTSKPOLB
SCHEMBL6509302 0.89 PDPK1 (0.41) PDPK1CTSKTSHRRECQLMEN1
SCHEMBL6512771 0.89 PDPK1 (0.44) PDPK1CTSKTSHRRECQLMEN1
SCHEMBL6530634 0.86 CTSK (0.45) CTSKALDH1A1HPGD
SCHEMBL6530210 0.85 NPC1 (0.45) CTSKTSHRKMT2ARAB9AKDM4E
SCHEMBL6530478 0.85 CTSK (0.43) CTSK
SCHEMBL6528746 0.84 CTSK (0.44) CTSKMEN1KMT2A
SCHEMBL6532662 0.84 CTSK (0.42) CTSKRECQLCYP2C9CYP2C19MMP1
SCHEMBL6530873 0.83 MAPT (0.41) CTSKTSHRMEN1KMT2AKDM4E
SCHEMBL6508189 0.83 KCNH3 (0.41) CTSKMEN1KMT2ACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO claimed