SCHEMBL6530826

SCHEMBL6530826

O=C(Nc1nc2cccc(O)c2n1CCN1CCOCC1)c1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.53
KDM4E B2RXH2 2/20 0.53
NPSR1 Q6W5P4 1/20 0.53
MTOR P42345 1/20 0.52
IRAK1 P51617 1/20 0.52
IRAK4 Q9NWZ3 1/20 0.52
TP53 P04637 2/20 0.49
HSD17B10 Q99714 2/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
RAB9A P51151 1/20 0.49
GAA P10253 2/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ROCK2 O75116 1/20 0.47
OPRK1 P41145 6/20 0.47
OPRM1 P35372 1/20 0.46
OPRD1 P41143 1/20 0.46
RPS6KA2 Q15349 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6505339 0.72 KDM4E (0.69) SMN1; SMN2KDM4ENPSR1MTORIRAK1
SCHEMBL16261073 0.71 MTOR (0.74) SMN1; SMN2KDM4ENPSR1MTORIRAK1
SCHEMBL5813832 0.71 SMN1; SMN2 (0.98) SMN1; SMN2KDM4EALDH1A1GAA
SCHEMBL2772319 0.70 SMN1; SMN2 (0.72) SMN1; SMN2TP53HSD17B10ALDH1A1GAA
SCHEMBL13500540 0.70 OPRK1 (0.86) SMN1; SMN2KDM4ENPSR1MTORIRAK1
SCHEMBL6530642 0.69 KDM4E (1.00) SMN1; SMN2KDM4ENPSR1MTORIRAK1
SCHEMBL3600001 0.69 MTOR (0.70) SMN1; SMN2KDM4ENPSR1MTORIRAK1
SCHEMBL28694253 0.69 SMN1; SMN2 (0.71) SMN1; SMN2TP53NPC1ALDH1A1RAB9A
SCHEMBL17554115 0.69 POLB (0.69) SMN1; SMN2ALDH1A1GAA
SCHEMBL3606266 0.69 CLK2 (0.72) KDM4ENPSR1MTORIRAK1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005021547-A2 HETEROCYCLIC CANNABINOID CB2 RECEPTOR ANTAGONISTS PHARMAXIS PTY LTD. (AU) 2005-03-10 WO disclosed