SCHEMBL6531002

SCHEMBL6531002

COc1ccc(CCNc2nc(Nc3cccc(F)c3)nc(N[C@@H](CO)CC(C)C)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CDK1 P06493 1/20 0.44
FCGR3B O75015 1/20 0.43
FCGR1A P12314 1/20 0.43
FCGR2A P12318 1/20 0.43
GBA1 P04062 2/20 0.43
IDH2 P48735 1/20 0.43
KCNH3 Q9ULD8 6/20 0.43
CNR2 P34972 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6531320 0.88 ALDH1A1 (0.45) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6530247 0.87 ALDH1A1 (0.47) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6530426 0.87 ALDH1A1 (0.47) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6530423 0.87 ALDH1A1 (0.47) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6530404 0.84 IDH2 (0.43) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6527570 0.84 IDH2 (0.43) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL6531883 0.83 KCNH3 (0.52) GBA1IDH2KCNH3
SCHEMBL13421323 0.80 FCGR3B (0.67) FCGR3BFCGR1AFCGR2AIDH2KCNH3
SCHEMBL6529521 0.79 IDH2 (0.47) IDH2KCNH3
SCHEMBL13421362 0.78 FCGR3B (0.61) FCGR3BFCGR1AFCGR2AIDH2KCNH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed