SCHEMBL6531737

SCHEMBL6531737

CC(C)CC(NC(=O)O)C(=O)NC(CCc1ccccc1)C(=O)C1=N[C@@H](c2ccccc2)CO1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 6/20 0.43
CTSS P25774 5/20 0.43
CTSB P07858 5/20 0.43
CTSK P43235 3/20 0.43
MMP3 P08254 4/20 0.42
REN P00797 1/20 0.41
MMP2 P08253 5/20 0.41
PSMB8 P28062 1/20 0.41
PSMB5 P28074 1/20 0.41
PSMB10 P40306 1/20 0.41
PSMB2 P49721 1/20 0.41
TMPRSS11D O60235 1/20 0.40
CTRL P40313 1/20 0.40
MMP1 P03956 2/20 0.40
ANPEP P15144 1/20 0.40
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6466342 0.90 CTSL (0.54) CTSLCTSSCTSBCTSK
SCHEMBL6466343 0.90 CTSL (0.54) CTSLCTSSCTSBCTSK
SCHEMBL7593794 0.80 CTSL (0.46) CTSLCTSSCTSB
SCHEMBL6468739 0.77 CTSL (0.54) CTSLCTSSCTSBCTSK
SCHEMBL6061622 0.77 CTSL (0.54) CTSLCTSSCTSBCTSK
SCHEMBL6467377 0.73 CTSL (0.54) CTSLCTSSCTSBCTSK
SCHEMBL7045967 0.72 SMN1; SMN2 (0.41)
SCHEMBL21457995 0.71 CAPN1 (0.64) CTSLCTSBMMP3RENMMP2
SCHEMBL3844110 0.71 CAPN1 (0.64) CTSLCTSBMMP3RENMMP2
SCHEMBL21458073 0.70 ANPEP (0.50) CTSLMMP3MMP2MMP1ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed