SCHEMBL6532226

SCHEMBL6532226

COc1ccc(Sc2cnc(Cl)nc2Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 2/20 0.44
DHFR P00374 1/20 0.44
HAO1 Q9UJM8 1/20 0.42
IDO1 P14902 1/20 0.42
POLB P06746 1/20 0.41
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PPP1CA P62136 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
SLC5A2 P31639 1/20 0.40
EGFR P00533 1/20 0.39
TYMS P04818 1/20 0.39
PDGFRB P09619 1/20 0.39
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
MMP12 P39900 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5408788 0.78 TP53 (0.48) MEN1KMT2AALDH1A1MAPTPOLB
SCHEMBL5861219 0.76 IDO1 (0.43) MEN1KMT2AALDH1A1MAPTDHFR
SCHEMBL17262275 0.75 MAOA (0.50) MEN1KMT2AALDH1A1MAPTDHFR
SCHEMBL7662525 0.73 HAO1 (0.46) MEN1KMT2AALDH1A1MAPTHAO1
SCHEMBL9044636 0.72 KMT2A (0.51) MEN1KMT2AMAPTHTT
SCHEMBL9150436 0.72 DHFR (0.60) KMT2ADHFRRXFP1EGFRTYMS
SCHEMBL30548759 0.72 MEN1 (0.62) MEN1KMT2AALDH1A1MAPTDHFR
SCHEMBL11392611 0.70 HAO1 (0.46) MEN1KMT2AALDH1A1MAPTDHFR
SCHEMBL829981 0.69 AURKA (0.48) MEN1KMT2AALDH1A1MAPTDHFR
SCHEMBL4692835 0.69 MAPT (0.45) MEN1KMT2AALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed