SCHEMBL9150436

SCHEMBL9150436

COc1ccc(Sc2cnc(N)nc2N)cc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 9/20 0.60
EGFR P00533 1/20 0.53
TYMS P04818 1/20 0.53
PDGFRB P09619 1/20 0.53
RXFP1 Q9HBX9 1/20 0.50
KMT2A Q03164 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9145080 0.79 RXFP1 (0.71) DHFREGFRTYMSRXFP1KMT2A
SCHEMBL19363998 0.76 P2RX3 (0.60) DHFR
SCHEMBL19407644 0.76 DHFR (0.50) DHFR
SCHEMBL13842554 0.72 P2RX3 (0.63) DHFRKMT2A
SCHEMBL30488020 0.72 KMT2A (0.73) DHFRKMT2A
SCHEMBL264291 0.72 KMT2A (0.73) DHFRKMT2A
SCHEMBL6532226 0.72 MEN1 (0.44) DHFREGFRTYMSPDGFRBRXFP1
SCHEMBL30548759 0.72 MEN1 (0.62) DHFREGFRTYMSPDGFRBKMT2A
SCHEMBL8964803 0.71 MEN1 (0.54) DHFREGFRTYMSPDGFRBKMT2A
SCHEMBL17097395 0.71 SMN1; SMN2 (0.54) DHFRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674627-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-10-04 EP disclosed
WO-1994014780-A1 PYRIMIDINE, PYRIDINE, PTERIDINONE AND INDAZOLE DERIVATIVES AS ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-07 WO disclosed