SCHEMBL6532351

SCHEMBL6532351

COC(=O)C(C)(Cc1ccc(OC(c2ccc(CC(C)C)cc2)c2cn[nH]c2)cc1)C(C)=NOCc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.32
ROCK2 O75116 2/20 0.32
ROCK1 Q13464 2/20 0.32
LTA4H P09960 1/20 0.32
PPARG P37231 7/20 0.31
PPARA Q07869 5/20 0.31
TSHR P16473 1/20 0.31
CTSL P07711 2/20 0.30
CTSB P07858 1/20 0.30
CTSF Q9UBX1 1/20 0.30
CTSK P43235 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6534135 0.93 PPARG (0.33) ACACBPPARGPPARACTSLCTSK
SCHEMBL6532684 0.83 PPARG (0.38) ACACBROCK2ROCK1LTA4HPPARG
SCHEMBL6532718 0.82 PPARG (0.43) PPARGPPARA
SCHEMBL6532377 0.76 PPARG (0.39) ROCK2ROCK1LTA4HPPARGPPARA
SCHEMBL6532102 0.76 PPARG (0.39) ROCK2ROCK1LTA4HPPARGPPARA
SCHEMBL6532609 0.76 PPARG (0.47) PPARGPPARA
SCHEMBL6533025 0.76 PPARG (0.40) PPARGPPARAMAOB
SCHEMBL6533825 0.76 PPARG (0.37) ROCK2LTA4HPPARGPPARA
SCHEMBL6533257 0.76 ROCK2 (0.34) ROCK2PPARGPPARAMAOB
SCHEMBL6532383 0.76 PPARG (0.40) ACACBROCK2ROCK1PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005040127-A1 NOVEL COMPOUNDS AS AGONIST FOR PPAR GAMMA AND PPAR ALPHA, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2005-05-06 WO claimed
WO-2005040127-A1 NOVEL COMPOUNDS AS AGONIST FOR PPAR GAMMA AND PPAR ALPHA, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2005-05-06 WO disclosed