SCHEMBL6532436

SCHEMBL6532436

O=C(C(O)CO)N1CCN(c2c(F)cc(C(c3c[nH]nn3)N3C(=O)c4ccccc4C3=O)cc2F)CC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RBP4 P02753 1/20 0.37
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.32
ALDH1A1 P00352 2/20 0.32
HTT P42858 1/20 0.32
GAA P10253 1/20 0.31
KMT2A Q03164 1/20 0.31
LMNA P02545 1/20 0.31
KDM4E B2RXH2 1/20 0.30
POLB P06746 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532785 0.91 RBP4 (0.40) RBP4NPC1TSHRALDH1A1HTT
SCHEMBL6532730 0.85 JAK3 (0.37) KMT2A
SCHEMBL6530631 0.78 MAPK1 (0.30)
SCHEMBL6527893 0.77 RBP4 (0.32) RBP4
SCHEMBL6530861 0.77 RBP4 (0.32) RBP4
SCHEMBL6533971 0.76 JAK3 (0.40) GAAKMT2A
SCHEMBL5623717 0.71 NPC1 (0.40) NPC1TSHRALDH1A1GAAKMT2A
SCHEMBL6532434 0.71 TYR (0.38) RBP4HTTGAAKMT2A
SCHEMBL6528273 0.69 CDK7 (0.39)
SCHEMBL6527385 0.69 RBP4 (0.39) RBP4TSHRALDH1A1HTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082892-A2 TRIAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S LABORATORIES LTD. (IN) 2005-09-09 WO disclosed