SCHEMBL6533971

SCHEMBL6533971

C=CC(=O)N1CCN(c2ccc(C(c3c[nH]nn3)N3C(=O)c4ccccc4C3=O)cc2F)CC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 4/20 0.40
KRAS P01116 7/20 0.38
GAA P10253 1/20 0.36
TET3 O43151 1/20 0.36
KMT2A Q03164 1/20 0.36
FBXL19 Q6PCT2 1/20 0.36
CXXC5 Q7LFL8 1/20 0.36
TET1 Q8NFU7 1/20 0.36
KDM2B Q8NHM5 1/20 0.36
CXXC4 Q9H2H0 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
EGFR P00533 3/20 0.35
KIT P10721 1/20 0.34
AURKB Q96GD4 1/20 0.34
SLC6A9 P48067 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532730 0.90 JAK3 (0.37) JAK3KRASTET3KMT2AFBXL19
SCHEMBL6532785 0.85 RBP4 (0.40) GAAKMT2ASLC6A9GPR55GRM5
SCHEMBL5623717 0.83 NPC1 (0.40) GAAKMT2A
SCHEMBL6527397 0.80 MAPK1 (0.35) GAAKMT2AGRM5
SCHEMBL6532436 0.76 RBP4 (0.37) GAAKMT2A
SCHEMBL6528273 0.72 CDK7 (0.39)
SCHEMBL6530631 0.71 MAPK1 (0.30)
SCHEMBL6533251 0.69 ALOX5AP (0.35)
SCHEMBL6346560 0.69 HPGD (0.39) KMT2A
SCHEMBL6925274 0.69 MAPK14 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082892-A2 TRIAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S LABORATORIES LTD. (IN) 2005-09-09 WO disclosed