SCHEMBL6534046

SCHEMBL6534046

CC(C)(C)c1ccc(-c2ccc(-c3cccnn3)c(Cl)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.42
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
XDH P47989 1/20 0.37
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
TRPV1 Q8NER1 2/20 0.35
CNR1 P21554 1/20 0.34
CCR9 P51686 1/20 0.34
PTAFR P25105 1/20 0.34
RAB9A P51151 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
NR2F2 P24468 1/20 0.33
DHODH Q02127 1/20 0.33
S1PR1 P21453 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23258136 0.78 KIF11 (0.50) KIF11XDHKMT2AALDH1A1KDM4E
SCHEMBL16013364 0.71 ALDH1A1 (0.44) ALDH1A1KDM4ERAB9ANPC1POLB
SCHEMBL18653354 0.71 HTR2C (0.35) KMT2AALDH1A1RAB9AMEN1NPC1
SCHEMBL29262131 0.71 KIF11 (0.41) KIF11KMT2AALDH1A1KDM4EDHODH
SCHEMBL14602201 0.69 AHR (0.61) KIF11AKR1C2AKR1C1XDHCNR1
SCHEMBL16780836 0.69 SLC6A2 (0.53) ALDH1A1KDM4ERAB9ANPC1DHODH
SCHEMBL15253926 0.68 RAB9A (0.46) KMT2AALDH1A1RAB9AMEN1NPC1
SCHEMBL19318451 0.68 DHODH (0.48) KIF11AKR1C2AKR1C1KMT2AALDH1A1
SCHEMBL10765944 0.68 IDO1 (0.46) ALDH1A1KDM4ERAB9ANPC1HPGD
SCHEMBL18653355 0.68 HTR2C (0.32) ALDH1A1RAB9ANPC1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542692-A1 AMINO-PYRIDINE, -PYRIDINE AND PYRIDAZINE DERIVATIVES FOR USE AS VANILLOID RECEPTOR LIGANDS FOR THE TREATMENT OF PAIN Amgen Inc. (US) 2005-06-22 EP disclosed
WO-2003099284-A1 AMINO-PYRIDINE, -PYRIDINE AND PYRIDAZINE DERIVATIVES FOR USE AS VANILLOID RECEPTOR LIGANDS FOR THE TREATMENT OF PAIN AMGEN INC. (US) 2003-12-04 WO disclosed