SCHEMBL6534667

SCHEMBL6534667

COC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.62
CASP3 P42574 2/20 0.59
CASP7 P55210 1/20 0.59
REN P00797 1/20 0.57
ALDH1A1 P00352 3/20 0.57
THRB P10828 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
HSD17B10 Q99714 1/20 0.57
CASP1 P29466 2/20 0.56
CASP9 P55211 1/20 0.56
MME P08473 1/20 0.55
ECE1 P42892 1/20 0.55
ALOX15 P16050 1/20 0.55
CAPN1 P07384 1/20 0.54
CTSD P07339 2/20 0.54
MDM4 O15151 1/20 0.54
MDM2 Q00987 1/20 0.54
CTSL P07711 2/20 0.53
CTSB P07858 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9416814 0.95 ALDH1A1 (0.62) TSHRCASP3ALDH1A1THRBCYP2C9
SCHEMBL8612642 0.92 ECE1 (0.64) CASP3CASP7RENCASP1CASP9
SCHEMBL28252140 0.92 ECE1 (0.64) CASP3CASP7RENCASP1CASP9
SCHEMBL8588834 0.91 ALDH1A1 (0.55) TSHRCASP3CASP7RENALDH1A1
SCHEMBL6271137 0.91 CASP3 (0.64) CASP3CASP7RENCASP1CASP9
SCHEMBL22413453 0.90 CASP3 (0.58) TSHRCASP3CASP7RENCASP1
SCHEMBL11211146 0.89 TSHR (0.57) TSHRALDH1A1THRBCYP2C9CYP2C19
SCHEMBL28607135 0.89 CASP3 (0.59) CASP3CASP7RENCASP1CASP9
SCHEMBL28607136 0.89 CASP3 (0.59) CASP3CASP7RENCASP1CASP9
SCHEMBL2402461 0.88 ALDH1A1 (0.67) TSHRALDH1A1THRBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828847-A4 ENZYME CATALYSIS IN ORGANIC SOLUTIONS BIOTECHNOLOGY RES & DEV (US) 2004-12-08 EP disclosed
US-6171813-B1 MIXING CATALYST OF ENZYME-SURFACTANT ION PAIR COMPLEX WITH ORGANIC REACTION SOLVENT INCLUDING WATER FROM 0.03 TO 2.5% V/V; WATER INCREASES RATE OF CATALYSIS AND STABILIZES ENZYME WITHOUT INCREASING RATE OF HYDROLYSIS; PEPTIDE SYNTHESIS BIOTECHNOLOGY RESEARCH & DEVELOP. CORP. 2001-01-09 US disclosed
EP-0828847-A1 ENZYME CATALYSIS IN ORGANIC SOLUTIONS BIOTECHNOLOGY RESEARCH AND DEVELOPMENT CORPORATION (US) 1998-03-18 EP disclosed
US-5719039-A FOR PEPTIDE SYNTHESIS FROM ACYL DONORS AND NUCLEOPHILES UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 1998-02-17 US disclosed
WO-1996038577-A1 ENZYME CATALYSIS IN ORGANIC SOLUTIONS BIOTECHNOLOGY RESEARCH AND DEVELOPMENT CORP. (US) 1996-12-05 WO disclosed