SCHEMBL6534968

SCHEMBL6534968

CC(CC(=O)O)(CC(=O)O)C(N)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.62
HIF1A Q16665 2/20 0.62
TSHR P16473 2/20 0.62
CYP2D6 P10635 1/20 0.62
HMGCR P04035 1/20 0.50
CHRM1 P11229 1/20 0.50
TBXA2R P21731 1/20 0.50
ADRA1A P35348 1/20 0.50
KDM4E B2RXH2 1/20 0.48
FFAR1 O14842 1/20 0.42
CPT2 P23786 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
FFAR3 O14843 1/20 0.33
GLRA1 P23415 1/20 0.33
SLC6A9 P48067 1/20 0.33
OR51E2 Q9H255 1/20 0.33
BHMT Q93088 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28001172 0.84 CYP2C19 (0.50) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL804144 0.78 KDM4E (0.54) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL503703 0.77 TSHR (1.00) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL28324214 0.74 CYP2C19 (0.65) CYP2C19HIF1ATSHRCYP2D6HMGCR
T-Butylacetic Acid SCHEMBL28024820 0.74 HMGCR (0.52) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL29020108 0.74 TSHR (0.94) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL6412305 0.74 CYP2C19 (0.50) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL11305042 0.74 CYP2C19 (0.71) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL27598677 0.72 HMGCR (0.44) CYP2C19HIF1ATSHRCYP2D6HMGCR
SCHEMBL9536247 0.71 HMGCR (0.55) CYP2C19HIF1ATSHRCYP2D6HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0941120-A4 BRANCHED PEPTIDE LINKERS BRISTOL MYERS SQUIBB CO (US) 2004-08-18 EP disclosed
EP-0941120-A1 BRANCHED PEPTIDE LINKERS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-09-15 EP disclosed
WO-1998019705-A1 BRANCHED PEPTIDE LINKERS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-14 WO disclosed