SCHEMBL6535170

SCHEMBL6535170

O=CNc1cccc(CCl)c1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
TSHR P16473 1/20 0.42
ADH1B P00325 1/20 0.35
ADH1C P00326 1/20 0.35
ADH1A P07327 1/20 0.35
ADH7 P40394 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
HTR6 P50406 1/20 0.33
EPHX1 P07099 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
LIMK1 P53667 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10133361 0.84 ALDH1A1 (0.52) ALDH1A1ADH1BADH1CADH1AADH7
SCHEMBL17383380 0.81 ALDH1A1 (0.48) ALDH1A1ADH1BADH1CADH1AADH7
SCHEMBL4598099 0.81 HTR6 (0.50) ALDH1A1HTR6
SCHEMBL19279237 0.81 ALDH1A1 (0.48) ALDH1A1TSHRADH1BADH1CADH1A
SCHEMBL1188674 0.81 RAPGEF4 (0.49) ALDH1A1GAAMAPT
SCHEMBL14401880 0.81 ALDH1A1 (0.48) ALDH1A1MAPT
SCHEMBL12129057 0.79 ALDH1A1 (0.67) ALDH1A1MAPTLIMK1
SCHEMBL11616567 0.78 CYP3A4 (0.50) ALDH1A1ADH1BADH1CADH1AADH7
SCHEMBL10388289 0.78 GRIN2D (0.47) ALDH1A1HTR6GAA
SCHEMBL13972907 0.77 SELP (0.52) ALDH1A1TSHRGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1237061-C Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2006-01-18 CN disclosed
EP-1242081-A4 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORP (US) 2004-07-21 EP disclosed
CN-1458929-A Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2003-11-26 CN disclosed
EP-1001933-A4 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORP (US) 2002-11-06 EP disclosed
EP-1242081-A1 CASPASES AND APOPTOSIS SmithKline Beecham Corporation (US) 2002-09-25 EP disclosed
WO-2001022966-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-05 WO disclosed
EP-1001933-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 2000-05-24 EP disclosed
WO-1999006367-A1 CASPASES AND APOPTOSIS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-11 WO disclosed