SCHEMBL6535453

SCHEMBL6535453

Oc1ccccc1CCc1ccccc1Sc1ccccc1CCc1ccccc1O

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.54
HSPA5 P11021 1/20 0.50
P4HB P07237 1/20 0.47
MPO P05164 4/20 0.47
CYP2D6 P10635 1/20 0.45
TSHR P16473 1/20 0.45
HIF1A Q16665 1/20 0.45
HTR1A P08908 1/20 0.44
SLC6A4 P31645 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
AKR1B1 P15121 1/20 0.43
IDO1 P14902 2/20 0.42
CA12 O43570 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29706272 0.83 TAAR1 (0.71) TAAR1HSPA5MPOCYP2D6TSHR
SCHEMBL1222973 0.83 TAAR1 (0.71) TAAR1HSPA5MPOCYP2D6TSHR
SCHEMBL29706378 0.81 TAAR1 (0.68) TAAR1HSPA5MPOCYP2D6TSHR
Ethane SCHEMBL10694585 0.79 TAAR1 (0.65) TAAR1HSPA5MPOCYP2D6TSHR
SCHEMBL588785 0.77 APOBEC3G (0.48) P4HBSLC6A4
Formaldehyde SCHEMBL28980606 0.77 TAAR1 (0.62) TAAR1HSPA5MPOCYP2D6TSHR
SCHEMBL25910731 0.76 HSPA5 (0.52) TAAR1HSPA5P4HBMPOCYP2D6
SCHEMBL12090255 0.75 P4HB (0.57) HSPA5P4HBCYP2D6TSHRSLC6A4
SCHEMBL4967651 0.74 TAAR1 (0.65) TAAR1HSPA5MPOCYP2D6TSHR
SCHEMBL3800530 0.74 TAAR1 (0.65) TAAR1HSPA5MPOCYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0958275-A4 SELECTIVE INHIBITORS OF PROSTAGLANDIN ENDOPEROXIDE SYNTHASE-2 UNIV VANDERBILT (US) 2004-12-01 EP disclosed
US-6284918-B1 ENZYME INHIBITORS VANDERBILT UNIVERSITY 2001-09-04 US disclosed
EP-0958275-A1 SELECTIVE INHIBITORS OF PROSTAGLANDIN ENDOPEROXIDE SYNTHASE-2 VANDERBILT UNIVERSITY (US) 1999-11-24 EP disclosed
US-5973191-A AN ACETOXYPHENYLALKYL SULFIDE, SALT OR HYDRATE VANDERBILT UNIVERSITY (US) 1999-10-26 US disclosed
WO-1998029382-A1 SELECTIVE INHIBITORS OF PROSTAGLANDIN ENDOPEROXIDE SYNTHASE-2 VANDERBILT UNIVERSITY (US) 1998-07-09 WO disclosed