SCHEMBL4276345

SCHEMBL4276345

COc1c(-c2ccccc2)cc(Cl)c(C=O)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PDE4B Q07343 3/20 0.41
PDE4A P27815 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
ERN1 O75460 1/20 0.41
CYP2A6 P11509 1/20 0.39
LCK P06239 1/20 0.39
GLA P06280 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
LIMK1 P53667 1/20 0.39
LIMK2 P53671 1/20 0.39
ACLY P53396 4/20 0.38
BACE1 P56817 3/20 0.37
IKBKB O14920 1/20 0.36
PTGS2 P35354 2/20 0.36
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10973832 0.88 ALDH1A1 (0.45) ALDH1A1KDM4EL3MBTL1PDE4BPDE4A
SCHEMBL29213635 0.80 MEN1 (0.42) ALDH1A1CYP2A6ACLYBACE1MEN1
SCHEMBL6535860 0.79 ALDH1A1 (0.49) ALDH1A1KDM4EL3MBTL1PDE4BPDE4A
SCHEMBL27812283 0.78 ALDH1A1 (0.41) ALDH1A1KDM4EL3MBTL1PDE4BPDE4A
SCHEMBL11051285 0.77 MEN1 (0.43) ALDH1A1KDM4EL3MBTL1PDE4BPDE4A
SCHEMBL17085611 0.77 ALDH1A1 (0.49) ALDH1A1KDM4EL3MBTL1PDE4BPDE4A
SCHEMBL881433 0.74 ERN1 (0.40) ALDH1A1KDM4EERN1MAPT
SCHEMBL6535962 0.72 ALDH1A1 (0.40) ALDH1A1KDM4EPDE4BPDE4APDE4C
SCHEMBL29672073 0.72 ERN1 (0.45) ALDH1A1KDM4EERN1LCKGLA
SCHEMBL6535983 0.72 ERN1 (0.45) ALDH1A1KDM4EERN1LCKGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2131655-A2 TRI-ARYL/HETEROAROMATIC CANNABINOIDS AND USE THEREOF The University of Tennessee Research Foundation (US) 2009-12-16 EP disclosed
WO-2008109027-A2 TRI-ARYL/HETEROAROAROMATIC CANNABINOIDS AND USE THEREOF UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION, THE (US) 2008-09-12 WO disclosed