SCHEMBL6536020

SCHEMBL6536020

COc1ccccc1-c1cccc(OC)c1C=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.47
TLR2 O60603 1/20 0.46
TLR1 Q15399 1/20 0.46
TLR6 Q9Y2C9 1/20 0.46
APP P05067 1/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
ALDH1A1 P00352 4/20 0.43
ABCG2 Q9UNQ0 1/20 0.42
HTR7 P34969 1/20 0.42
UGCG Q16739 1/20 0.42
TOP1 P11387 1/20 0.42
KDM4E B2RXH2 2/20 0.41
USP2 O75604 2/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3679777 0.87 ERN1 (0.54) ERN1TLR2TLR1TLR6CA1
SCHEMBL9754385 0.85 ERN1 (0.45) ERN1TLR2TLR1TLR6CA12
SCHEMBL6536507 0.85 ALDH1A1 (0.48) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL170690 0.83 ERN1 (0.55) ERN1TLR2TLR1TLR6CA12
SCHEMBL27685686 0.79 ERN1 (0.52) ERN1TLR2TLR1TLR6CA12
Bromomethane SCHEMBL28079811 0.79 ERN1 (0.52) ERN1TLR2TLR1TLR6CA12
SCHEMBL7932563 0.79 ERN1 (0.44) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL17597905 0.79 NFE2L2 (0.42) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL29912323 0.79 NFE2L2 (0.42) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL2474418 0.78 ERN1 (0.57) ERN1TLR2TLR1TLR6APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425015-A4 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2004-12-15 EP disclosed
EP-1425015-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-09 EP disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed