SCHEMBL6536174

SCHEMBL6536174

COc1ccc(-c2ccccc2)c(C(=O)O)c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
HK2 P52789 1/20 0.49
MAPT P10636 5/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
ALOX15 P16050 1/20 0.47
MAPK1 P28482 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDO2 P48775 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ERN1 O75460 3/20 0.43
ALDH1A1 P00352 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6535999 0.87 HK2 (0.56) CA12CA1CA2CA7CA9
SCHEMBL8381595 0.83 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL28667937 0.83 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL14322385 0.82 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL21638050 0.81 TDO2 (0.47) HK2MAPTMEN1KMT2AKDM4E
SCHEMBL4063174 0.80 CA12 (0.55) CA12CA1CA2CA7CA9
SCHEMBL9064266 0.80 CA12 (0.63) CA12CA1CA2CA7CA9
SCHEMBL4002652 0.79 CA12 (0.69) CA12CA1CA2CA7CA9
SCHEMBL30536599 0.79 CA12 (0.69) CA12CA1CA2CA7CA9
SCHEMBL30393914 0.79 CA12 (0.53) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425015-A4 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2004-12-15 EP disclosed
EP-1425015-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-09 EP disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed