SCHEMBL6537056

SCHEMBL6537056

CNc1cc(C)c(Nc2ccccc2)c2c1C(=O)OC21c2ccccc2Oc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.40
ALDH1A1 P00352 3/20 0.40
ALOX12 P18054 2/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
BRCA1 P38398 1/20 0.40
HSD17B10 Q99714 1/20 0.40
FTO Q9C0B1 4/20 0.34
MAPT P10636 4/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
BLM P54132 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
HTT P42858 2/20 0.34
CYP2C19 P33261 1/20 0.34
RECQL P46063 1/20 0.34
SMAD3 P84022 1/20 0.34
PRMT1 Q99873 1/20 0.34
ACE2 Q9BYF1 1/20 0.34
CXCR2 P25025 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11003355 0.89 HPGD (0.39) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL9565549 0.89 HPGD (0.38) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL2185607 0.86 ALDH1A1 (0.41) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL548194 0.85 CYP2C9 (0.36) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL10885589 0.85 HPGD (0.40) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL339448 0.84 TLR8 (0.36) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL395637 0.84 ALDH1A1 (0.35) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL4077129 0.84 ALDH1A1 (0.35) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL11039571 0.84 HSD17B10 (0.35) HPGDALDH1A1ALOX12CYP2C9ALOX15
SCHEMBL4667092 0.84 CYP2C9 (0.39) HPGDALDH1A1ALOX12CYP2C9ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6740465-B2 MULTILAYER; TRANSPARENT SUPPORT; HEAT SENSITIVE ELEMENT AND RELEASE AGENT SIPIX IMAGING, INC. 2004-05-25 US disclosed
EP-1289768-A2 IMAGING MEDIA CONTAINING HEAT DEVELOPABLE PHOTOSENSITIVE MICROCAPSULES Sipix Imaging, Inc. (US) 2003-03-12 EP disclosed
US-20020155372-A1 Imaging media containing heat developable photosensitive microcapsules SIPIX IMAGING, INC. 2002-10-24 US disclosed
US-20020065197-A1 Heat sensitive recording material LIANG RONG-CHANG (US) 2002-05-30 US disclosed
WO-2001092024-A2 IMAGING MEDIA CONTAINING HEAT DEVELOPABLE PHOTOSENSITIVE MICROCAPSULES SIPIX IMAGING, INC. (US) 2001-12-06 WO disclosed
US-6326071-B1 Reverse thermal label NASHUA CORPORATION 2001-12-04 US disclosed
WO-2001054917-A1 HEAT SENSITIVE RECORDING MATERIAL SIPIX IMAGING, INC. (US) 2001-08-02 WO disclosed
US-6107244-A Verification methods employing thermally--imageable substrates NASHUA CORPORATION (US) 2000-08-22 US disclosed
EP-0942835-A1 VERIFICATION METHODS AND SYSTEMS EMPLOYING THERMALLY-IMAGEABLE SUBSTRATES NASHUA CORPORATION (US) 1999-09-22 EP disclosed
WO-1999019150-A1 VERIFICATION METHODS AND SYSTEMS EMPLOYING THERMALLY-IMAGEABLE SUBSTRATES NASHUA CORPORATION (US) 1999-04-22 WO disclosed
US-5219821-A Friction reducing protective layer of organic water soluble resin crosslinked in situ with nonacidic crosslinking agent, inorganic nonacidic filler NASHUA CORPORATION (US) 1993-06-15 US disclosed
WO-1992014615-A1 NON-ACIDIC BARRIER COATING NASHUA CORPORATION (US) 1992-09-03 WO disclosed
US-5141914-A Crosslinked binder protective coating NASHUA CORPORATION (US) 1992-08-25 US disclosed
US-5075369-A Mixture of curable resin, ionic and covalent crosslinking agents, acid catalyst forms solvent resistant protective coating having discoloration resistance NASHUA CORPORATION (US) 1991-12-24 US disclosed
EP-0355146-A4 COATED THERMALLY PRINTABLE MATERIAL AND METHOD OF PRODUCING THE SAME 1991-05-22 EP disclosed
US-4927801-A HEAT SENSITIVE RECORDING MATERIAL NASHUA CORPORATION (US) 1990-05-22 US disclosed
EP-0355146-A1 COATED THERMALLY PRINTABLE MATERIAL AND METHOD OF PRODUCING THE SAME NASHUA CORPORATION (US) 1990-02-28 EP disclosed
US-4898849-A PROTECTIVE COATING OF CROSS-LINKED RESIN, FRICTION-REDUCTING POLYMER PARTICLE AND FLUOROCARBON SURFACTANT; SOLVENT-RESISTANT, COLORFAST LABELS; FOOD APPARATUS NASHUA CORPORATION (US) 1990-02-06 US disclosed
WO-1989006191-A1 COATED THERMALLY PRINTABLE MATERIAL AND METHOD OF PRODUCING THE SAME NASHUA CORPORATION (US) 1989-07-13 WO disclosed