SCHEMBL6539799

SCHEMBL6539799

COc1ccc(-c2nc(C(C)C)oc2-c2ccc(OCCN)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
MAPT P10636 3/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
POLB P06746 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
DHFR P00374 1/20 0.39
PPARD Q03181 5/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
MAOB P27338 1/20 0.35
DPP4 P27487 1/20 0.35
KDR P35968 1/20 0.35
TEK Q02763 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
CASP1 P29466 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6539783 0.89 ALDH1A1 (0.39) ALDH1A1MAPTKDM4EHPGDPOLB
SCHEMBL6539669 0.89 KDM4E (0.41) ALDH1A1MAPTKDM4EHPGDPOLB
Hydrochloric Acid SCHEMBL6207772 0.88 KMT2A (0.39) ALDH1A1MAPTKDM4EHPGDPOLB
Hydrochloric Acid SCHEMBL6539698 0.88 KMT2A (0.39) ALDH1A1MAPTKDM4EHPGDPOLB
SCHEMBL6539388 0.88 PPARD (0.38) PPARDKMT2AMEN1
SCHEMBL6258696 0.84 PPARD (0.40) ALDH1A1MAPTKDM4EHPGDPOLB
SCHEMBL6255182 0.83 PPARD (0.37) ALDH1A1MAPTKDM4EHPGDPOLB
SCHEMBL6231402 0.82 MTNR1A (0.45) ALDH1A1KDM4EHPGDPPARDKMT2A
SCHEMBL6540424 0.81 ALDH1A1 (0.42) ALDH1A1MAPTKDM4EHPGDPOLB
SCHEMBL6538937 0.81 NPSR1 (0.51) ALDH1A1MAPTKDM4EHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040157891-A1 Inhibitor of cox FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-08-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040157891-A1 Inhibitor of cox PTGS1, PTGS2, PTGES2 ALDH1A1 163/4885MAPT 4796/4885KDM4E 1912/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.