SCHEMBL6540417

SCHEMBL6540417

CC(N)Oc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc3c(c2)OCO3)cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.57
PTGS1 P23219 8/20 0.53
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
THPO P40225 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
HIF1A Q16665 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5147766 0.82 PTGS2 (0.57) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL7472447 0.80 PTGS2 (0.60) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL7467786 0.79 PTGS2 (0.70) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL5152237 0.76 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL5147903 0.75 PTGS2 (0.52) PTGS2PTGS1CYP2C9
SCHEMBL5148844 0.74 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6343314 0.73 PTGS2 (1.00) PTGS2PTGS1CYP3A4CYP2C9TSHR
SCHEMBL7112386 0.70 PTGS2 (1.00) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL7468667 0.70 PTGS2 (0.71) PTGS2PTGS1CYP2C9
SCHEMBL6166763 0.69 PTGS2 (0.67) PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116475-A1 Pyrazole derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-06-17 US disclosed