SCHEMBL6541508

SCHEMBL6541508

CCOc1ccc(C=NO)c(F)c1-c1cc2c(cc1C)C(C)(C)CCC2(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.41
TSHR P16473 2/20 0.41
RXRA P19793 10/20 0.36
HNF4A P41235 5/20 0.36
RXRG P48443 5/20 0.35
RXRB P28702 3/20 0.35
RARA P10276 2/20 0.35
RARB P10826 2/20 0.35
RARG P13631 2/20 0.35
PKM P14618 1/20 0.35
GAA P10253 2/20 0.34
PDK2 Q15119 1/20 0.34
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6541500 1.00 HPGD (0.41) HPGDTSHRRXRAHNF4ARXRG
SCHEMBL6541989 0.88 RXRA (0.35) HPGDRXRARXRGRXRBRARA
SCHEMBL6541992 0.88 RXRA (0.35) HPGDRXRARXRGRXRBRARA
SCHEMBL7053364 0.84 RXRA (0.34) HPGDTSHRRXRAHNF4ARXRG
SCHEMBL7053359 0.84 RXRA (0.34) HPGDTSHRRXRAHNF4ARXRG
SCHEMBL6541475 0.82 RXRA (0.43) RXRARXRGRXRBRARARARB
SCHEMBL6541470 0.82 RXRA (0.43) RXRARXRGRXRBRARARARB
SCHEMBL6542800 0.78 GAA (0.46) HPGDTSHRRXRAHNF4ARXRG
SCHEMBL6542802 0.78 GAA (0.46) HPGDTSHRRXRAHNF4ARXRG
SCHEMBL5493911 0.78 IGF1R (0.47) HPGDRXRAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421061-A4 OXIME DERIVATIVES FOR THE TREATMENT OF DYSLIPIDEMIA AND HYPERCHOLESTEREMIA INCYTE SAN DIEGO INC (US) 2004-12-22 EP disclosed
EP-1421061-A1 OXIME DERIVATIVES FOR THE TREATMENT OF DYSLIPIDEMIA AND HYPERCHOLESTEREMIA Incyte San Diego Incorporated (US) 2004-05-26 EP disclosed
US-20030083357-A1 Oxime derivatives for the treatment of dyslipidemia and hypercholesteremia ORTHO MCNEIL PHARMACEUTICAL INC. 2003-05-01 US disclosed
WO-2003016267-A1 OXIME DERIVATIVES FOR THE TREATMENT OF DYSLIPIDEMIA AND HYPERCHOLESTEREMIA INCYTE SAN DIEGO INCORPORATED (US) 2003-02-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030083357-A1 Oxime derivatives for the treatment of dyslipidemia and hypercholesteremia OAT, CPT1A, CYP27A1 HPGD 524/4885TSHR 974/4885RXRA 793/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.