SCHEMBL6542722

SCHEMBL6542722

O=C(O)OC1=C(O)c2ccccc2S(=O)(=O)N1c1ccccc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.38
HSD11B1 P28845 2/20 0.38
LMNA P02545 1/20 0.36
MAPT P10636 3/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CA12 O43570 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 1/20 0.35
KDM4E B2RXH2 2/20 0.34
USP2 O75604 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX15 P16050 1/20 0.34
NFKB1 P19838 1/20 0.34
PTGS1 P23219 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6541894 0.85 ELANE (0.38) ELANEHSD11B1LMNAMAPTCA12
SCHEMBL6542043 0.84 HSD11B1 (0.36) ELANEHSD11B1LMNAMAPTTP53
SCHEMBL6542189 0.81 HSD11B1 (0.42) ELANEHSD11B1LMNAMAPTCA12
SCHEMBL6542021 0.78 MAPT (0.40) MAPTCA12CA9KDM4ECYP1A2
SCHEMBL6542499 0.77 HSD11B1 (0.47) ELANEHSD11B1LMNAKDM4EUSP2
SCHEMBL6541959 0.74 EDNRA (0.40) HSD11B1LMNAUSP2HPGD
SCHEMBL6542556 0.74 EDNRA (0.37) HSD11B1LMNASMN1; SMN2KDM4EHPGD
SCHEMBL6542004 0.74 HSD11B1 (0.45) ELANEHSD11B1LMNAMAPTTP53
SCHEMBL6542551 0.72 LMNA (0.65) ELANELMNASMN1; SMN2CA12CA2
SCHEMBL6542020 0.71 EDNRA (0.49) LMNAMAPTSMN1; SMN2KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1009743-B1 CERTAIN BENZOTHIAZINE DIOXIDE ENDOTHELIN ANTAGONISTS AND PROCESSES FOR THEIR PREPARATION WARNER LAMBERT CO (US) 2004-06-30 EP claimed