SCHEMBL654532

SCHEMBL654532

O=C(c1ccc(Cl)cc1)C1CCNCC1

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
CYP2D6 P10635 1/20 0.67
MGLL Q99685 10/20 0.58
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
MAPT P10636 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HSD11B1 P28845 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL229430 0.98 MEN1 (0.70) MEN1KMT2ACYP2D6MGLLLMNA
SCHEMBL13391197 0.87 MGLL (0.65) MEN1KMT2AMGLLHSD11B1
(4-Chlorophenyl)(Cyclopropyl)Methanone SCHEMBL392801 0.86 MGLL (0.68) MEN1KMT2AMGLLLMNATP53
SCHEMBL11354827 0.85 MEN1 (0.54) MEN1KMT2ACYP2D6MGLLLMNA
SCHEMBL8106011 0.85 MGLL (0.58) MEN1KMT2AMGLLLMNATP53
Tert-Butyl Formate SCHEMBL28875402 0.84 MEN1 (0.54) MEN1KMT2ACYP2D6MGLLLMNA
Hydrochloric Acid SCHEMBL11355129 0.84 MEN1 (0.56) MEN1KMT2ACYP2D6MGLLLMNA
SCHEMBL13944266 0.83 MEN1 (0.69) MEN1KMT2ACYP2D6TP53HSD11B1
SCHEMBL13390936 0.83 MEN1 (0.54) MEN1KMT2ACYP2D6MGLL
SCHEMBL5218517 0.83 MEN1 (0.69) MEN1KMT2ACYP2D6MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 224 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240016775-A1 ANTI-CORONAVIRUS APPLICATION OF POLY ADP RIBOSE POLYMERASE INHIBITOR FUKANG (SHANGHAI) HEALTH TECHNOLOGY CO., LTD (CN) 2024-01-18 US disclosed
US-20230015617-A1 PHTHALAZINONE DERIVATIVES KUDOS PHARMACEUTICALS LIMITED (GB) 2023-01-19 US disclosed
EP-3265453-B1 NEW PYRIDINONES AND ISOQUINOLINONES AS INHIBITORS OF THE BROMODOMAIN BRD9 BOEHRINGER INGELHEIM INT (DE) 2022-06-29 EP disclosed
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2022-05-03 US disclosed
US-11160803-B2 Phthalazinone derivatives KUDOS PHARMACEUTICALS LIMITED (GB) 2021-11-02 US disclosed
CN-106946796-B Aminopyrimidine derivatives useful as modulators of kinase activity 默克专利有限公司 2020-05-08 CN disclosed
US-10449192-B2 Phthalazinone derivatives KUDO PHARMACEUTICALS LIMITED (GB) 2019-10-22 US disclosed
WO-2019072978-A1 MITOCHONDRIAL INHIBITORS FOR THE TREATMENT OF PROLIFERATION DISORDERS Basilea Pharmaceutica International AG (CH) 2019-04-18 WO disclosed
US-10080750-B2 Aminopyrimidine derivatives for use as modulators of kinase activity MERCK PATENT GMBH (DE) 2018-09-25 US disclosed
US-RE46942-E1 4-piperidinyl compounds for use as tankyrase inhibitors NOVARTIS AG (CH) 2018-07-10 US disclosed
US-5232924-A Cardiovascular disorders DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1993-08-03 US disclosed
US-5206239-A Cardiovascular disorders SUNTORY LIMITED (JP) 1993-04-27 US disclosed
EP-0441349-A1 Pyrroloazepine derivatives SUNTORY LIMITED (JP) 1991-08-14 EP disclosed
US-4983606-A Pharmaceutically-active phthalazine compounds ZAMBON GROUP S.P.A. (IT) 1991-01-08 US disclosed
EP-0401707-A1 Heterocyclic triazin or triazolo compounds having serotonin 2-receptor antagonistic activity DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1990-12-12 EP disclosed
EP-0124476-B1 CARBOXAMIDES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM CIBA-GEIGY AG (CH) 1988-06-22 EP disclosed
US-4559349-A TREATMENT OF PHYCHOSIS CIBA GEIGY CORPORATION (US) 1985-12-17 US disclosed
EP-0124476-A1 Carboxamides, process for their preparation and pharmaceutical preparations containing them CIBA-GEIGY AG (CH) 1984-11-07 EP disclosed
US-4101662-A DISUBSTITUTED PIPERIDINES A. H. ROBINS COMPANY, INCORPORATED (US) 1978-07-18 US disclosed
US-3968217-A ANTIDEPRESSANT A. H. ROBINS COMPANY, INCORPORATED (US) 1976-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10080750-B2 Aminopyrimidine derivatives for use as modulators of kinase activity CDK6, TK1, MAP3K19 MEN1 3016/4885KMT2A 643/4885CYP2D6 2536/4885
US-10449192-B2 Phthalazinone derivatives NR0B1, NR0B2, NR2E1 MEN1 1409/4885KMT2A 2203/4885CYP2D6 1407/4885
US-11160803-B2 Phthalazinone derivatives NR0B1, NR0B2, NR2E1 MEN1 1409/4885KMT2A 2203/4885CYP2D6 1407/4885
US-20240016775-A1 ANTI-CORONAVIRUS APPLICATION OF POLY ADP RIBOSE POLYMERASE INHIBITOR PARP3, PARP1, PARP4 MEN1 4478/4885KMT2A 2392/4885CYP2D6 3250/4885
US-11319318-B2 Pyridinones and isoquinolinones as inhibitors of the bromodomain BRD9 BRD9, BRD1, BRD2 MEN1 1532/4885KMT2A 1279/4885CYP2D6 1852/4885
US-20230015617-A1 PHTHALAZINONE DERIVATIVES NR0B1, NR0B2, NR2E1 MEN1 1419/4885KMT2A 2142/4885CYP2D6 1395/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.