SCHEMBL6546249

SCHEMBL6546249

COc1c(Cc2cc(F)c3[nH]nc(-c4ccc5ccccc5c4)c3c2)cccc1C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.38
CDK4 P11802 2/20 0.37
CCND1 P24385 2/20 0.37
CDK2 P24941 2/20 0.37
CCNA2 P20248 1/20 0.37
CCND3 P30281 1/20 0.37
KDR P35968 1/20 0.37
GPR52 Q9Y2T5 1/20 0.36
CCNE2 O96020 1/20 0.35
CCNE1 P24864 1/20 0.35
PARP10 Q53GL7 3/20 0.35
PARP15 Q460N3 2/20 0.35
PDE10A Q9Y233 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
ALPL P05186 1/20 0.34
PARP14 Q460N5 1/20 0.34
CD38 P28907 1/20 0.33
NPY5R Q15761 1/20 0.33
CHEK2 O96017 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860995 0.76 HPGD (0.47) CDK4CCND1CDK2CCNA2CCND3
SCHEMBL2869259 0.74 MAPK8 (0.39) CDK4CCND1CDK2CCNA2CCND3
SCHEMBL2872869 0.73 ROCK2 (0.50) LMNAGSK3B
SCHEMBL13636075 0.70 CDK4 (0.47) PARP1CDK4CCND1CDK2CCNA2
SCHEMBL2865008 0.69 CSNK1D (0.44) KDRCHEK2JAK2
SCHEMBL2861275 0.69 CA12 (0.50) CDK4CCND1CDK2CCNA2CCND3
SCHEMBL2864472 0.68 IKBKB (0.43) CDK4CCND1CDK2CCNA2CCND3
SCHEMBL2867285 0.67 ITK (0.45) CDK4CCND1CDK2CCNA2CCND3
SCHEMBL4334282 0.66 SCN9A (0.39) CDK4CCND1CDK2CCNA2CCND3
SCHEMBL2870025 0.66 ROCK2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1380576-A1 NOVEL 1H-INDAZOLE COMPOUND Eisai Co., Ltd. (JP) 2004-01-14 EP disclosed