SCHEMBL6548168

SCHEMBL6548168

C#CS(=O)(=O)c1c(C)cc(C)cc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 3/20 0.47
PRSS1 P07477 3/20 0.47
PRSS2 P07478 3/20 0.47
PRSS3 P35030 3/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
MMP1 P03956 1/20 0.47
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
MMP13 P45452 1/20 0.47
RAPGEF4 Q8WZA2 6/20 0.45
NPSR1 Q6W5P4 1/20 0.44
GAA P10253 3/20 0.38
POLB P06746 2/20 0.38
TSHR P16473 2/20 0.38
GFER P55789 1/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6548063 0.74 RAPGEF4 (0.47) F2PRSS1PRSS2PRSS3CA1
SCHEMBL21117641 0.72 CA1 (0.56) F2PRSS1PRSS2PRSS3CA1
SCHEMBL2047218 0.72 RAPGEF4 (0.67) F2PRSS1PRSS2PRSS3CA1
SCHEMBL9803133 0.71 F2 (0.61) F2PRSS1PRSS2PRSS3CA1
SCHEMBL7458962 0.70 ALDH1A1 (0.36) F2PRSS1PRSS2PRSS3CA1
SCHEMBL330754 0.70 CA1 (0.54) F2PRSS1PRSS2PRSS3CA1
SCHEMBL8271353 0.70 CA1 (0.54) F2PRSS1PRSS2PRSS3CA1
SCHEMBL14516136 0.70 F2 (0.59) F2PRSS1PRSS2PRSS3CA1
SCHEMBL31066637 0.70 CA1 (0.53) F2PRSS1PRSS2PRSS3CA1
SCHEMBL16140087 0.70 F2 (0.53) F2PRSS1PRSS2PRSS3CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1162962-B1 ALKYNYL ARYL SULFONES LONZA AG (US) 2004-12-01 EP disclosed
EP-1162962-A4 ALKYNYL ARYL SULFONES LONZA AG (US) 2002-10-30 EP disclosed
EP-1162962-A1 ALKYNYL ARYL SULFONES LONZA INC. (US) 2001-12-19 EP disclosed
US-6232503-B1 MICROBIOCIDES LONZA INC. 2001-05-15 US disclosed
WO-2000056305-A1 ALKYNYL ARYL SULFONES LONZA INC. (US) 2000-09-28 WO disclosed