SCHEMBL6553355

SCHEMBL6553355

CCOC(=O)/C=C(/C)c1cc(Br)cc(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.43
MAPT P10636 5/20 0.41
LMNA P02545 4/20 0.41
F2 P00734 1/20 0.40
PLG P00747 1/20 0.40
PRSS1 P07477 1/20 0.40
GPR35 Q9HC97 1/20 0.40
ALDH1A1 P00352 4/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
S1PR4 O95977 1/20 0.38
S1PR1 P21453 1/20 0.38
MAPK1 P28482 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38
GALK1 P51570 1/20 0.38
CCR6 P51684 1/20 0.38
BLM P54132 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6553357 1.00 NPSR1 (0.43) NPSR1MAPTLMNAF2PLG
SCHEMBL29866648 0.89 XPO1 (0.41) NPSR1MAPTLMNAF2PLG
SCHEMBL2192541 0.85 KMT2A (0.47) NPSR1MAPTLMNAF2PLG
SCHEMBL2192534 0.85 KMT2A (0.47) NPSR1MAPTLMNAF2PLG
SCHEMBL2192538 0.85 KMT2A (0.47) NPSR1MAPTLMNAF2PLG
SCHEMBL4145995 0.84 ALDH1A1 (0.50) NPSR1MAPTLMNAF2PLG
SCHEMBL30152652 0.84 ALDH1A1 (0.50) NPSR1MAPTLMNAF2PLG
SCHEMBL4145986 0.84 ALDH1A1 (0.50) NPSR1MAPTLMNAF2PLG
SCHEMBL4145990 0.84 ALDH1A1 (0.50) NPSR1MAPTLMNAF2PLG
SCHEMBL6555579 0.82 RXRA (0.45) NPSR1MAPTALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1149067-B1 7-ARYL-6(Z)HEPTATRIENOIC ACID RETINAMIDES AS APOPTOSIS INDUCING COMPOUNDS AND THEIR USE AS ANTI-CANCER AGENTS HOFFMANN LA ROCHE (CH) 2004-02-25 EP disclosed
EP-1149067-A1 7-ARYL-6(Z)HEPTATRIENOIC ACID RETINAMIDES AS APOPTOSIS INDUCING COMPOUNDS AND THEIR USE AS ANTI-CANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2001-10-31 EP disclosed
US-6310247-B1 HAS APOPTOTIC ACTIVITY USEFUL FOR PROPHYLAXIS AND THERAPY OF CANCER HOFFMANN-LA ROCHE INC. 2001-10-30 US disclosed
WO-2000035856-A1 7-ARYL-6(Z)HEPTATRIENOIC ACID RETINAMIDES AS APOPTOSIS INDUCING COMPOUNDS AND THEIR USE AS ANTI-CANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed