SCHEMBL6555532

SCHEMBL6555532

COc1ccc(F)cc1C1(CC(=O)C(=O)O)CC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.43
HTR2C P28335 3/20 0.43
HTR2B P41595 2/20 0.43
PIN1 Q13526 3/20 0.41
KMT2A Q03164 2/20 0.39
HTT P42858 2/20 0.39
FFAR4 Q5NUL3 3/20 0.39
AKR1B1 P15121 2/20 0.39
FFAR1 O14842 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6554293 0.83 HTT (0.54) KMT2AHTTSMN1; SMN2KDM4EALDH1A1
SCHEMBL1633723 0.83 HTR2A (0.42) HTR2AHTR2CHTR2BPIN1KMT2A
SCHEMBL27687662 0.81 HTT (0.42) PIN1KMT2AHTTALDH1A1
SCHEMBL4826643 0.76 ALDH1A1 (0.41) KMT2AAKR1B1KDM4EALDH1A1MAPK1
SCHEMBL1262117 0.73 HDAC4 (0.35) KMT2AHTTKDM4EALDH1A1
SCHEMBL6554195 0.72 NR3C1 (0.53) KDM4EALDH1A1
SCHEMBL5643865 0.71 P2RX7 (0.43) AKR1B1ALDH1A1
SCHEMBL4816885 0.71 NR3C1 (0.40) HTR2AHTR2CHTR2BPIN1
SCHEMBL30040332 0.71 HTT (0.67) KMT2AHTTSMN1; SMN2KDM4EALDH1A1
SCHEMBL1634501 0.70 ALDH1A1 (0.43) HTR2AHTR2CHTR2BPIN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133486-B1 NONSTEROIDAL ANTIINFLAMMATORIES SCHERING AG (DE) 2004-12-22 EP disclosed
US-6323199-B1 AROMATIC HETEROCYCLIC HYDROXY AMINES OR AMIDES FOR TREATMENT OF INFLAMMATION SCHERING AKTIENGESELLSCHAFT (DE) 2001-11-27 US disclosed
EP-1133486-A2 NONSTEROIDAL ANTIINFLAMMATORIES SCHERING AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032584-A2 NONSTEROIDAL ANTIINFLAMMATORIES SCHERING AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed