SCHEMBL6558013

SCHEMBL6558013

O=[N+]([O-])c1ccc2nc(N3CC4CCCCCCCCCCCCCCCCCCCCCC3CC4)ccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
HTR3E A5X5Y0 1/20 0.49
HTR3B O95264 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
SLC6A4 P31645 1/20 0.49
CYP2C19 P33261 1/20 0.49
THPO P40225 1/20 0.49
HTR3A P46098 1/20 0.49
HTR3D Q70Z44 1/20 0.49
HTR3C Q8WXA8 1/20 0.49
HTR1A P08908 7/20 0.44
LMNA P02545 1/20 0.43
PMP22 Q01453 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MCHR1 Q99705 1/20 0.42
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5873479 0.94 ALDH1A1 (0.54) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL6559990 0.80 MCHR1 (0.43) ALDH1A1LMNAMCHR1NPC1POLB
SCHEMBL3386080 0.78 ALDH1A1 (0.58) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL3540666 0.78 ALDH1A1 (0.60) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL4846555 0.77 ALDH1A1 (0.51) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL27480804 0.75 ALDH1A1 (0.57) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL5832121 0.74 ALDH1A1 (0.59) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL4848007 0.74 ALDH1A1 (0.53) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4
SCHEMBL5873493 0.73 MCHR1 (0.46) ALDH1A1SLC6A4HTR3AHTR1ALMNA
SCHEMBL5873582 0.73 ALDH1A1 (0.76) ALDH1A1HTR3EHTR3BCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450801-A2 2-AMINOQUINOLINE COMPOUNDS Merck & Co., Inc. (US) 2004-09-01 EP disclosed
WO-2003045313-A2 2-AMINOQUINOLINE COMPOUNDS MERCK & CO. INC. (US) 2003-06-05 WO disclosed